Development of Potent and Selective Agonists for Complement C5a Receptor 1 with In Vivo Activity.

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Title: Development of Potent and Selective Agonists for Complement C5a Receptor 1 with In Vivo Activity.
Authors: Gorman DM; School of Biomedical Sciences, The University of Queensland, Brisbane, Queensland 4072, Australia., Li XX; School of Biomedical Sciences, The University of Queensland, Brisbane, Queensland 4072, Australia., Lee JD; School of Biomedical Sciences, The University of Queensland, Brisbane, Queensland 4072, Australia., Fung JN; School of Biomedical Sciences, The University of Queensland, Brisbane, Queensland 4072, Australia., Cui CS; School of Biomedical Sciences, The University of Queensland, Brisbane, Queensland 4072, Australia., Lee HS; School of Biomedical Sciences, The University of Queensland, Brisbane, Queensland 4072, Australia., Rolfe BE; Australian Institute for Bioengineering and Nanotechnology, The University of Queensland, Brisbane, Queensland 4072, Australia., Woodruff TM; School of Biomedical Sciences, The University of Queensland, Brisbane, Queensland 4072, Australia.; Queensland Brain Institute, The University of Queensland, Brisbane, Queensland 4072, Australia., Clark RJ; School of Biomedical Sciences, The University of Queensland, Brisbane, Queensland 4072, Australia.
Source: Journal of medicinal chemistry [J Med Chem] 2021 Nov 25; Vol. 64 (22), pp. 16598-16608. Date of Electronic Publication: 2021 Nov 11.
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: Development of Potent and Selective Agonists for Complement C5a Receptor 1 with In Vivo Activity.
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  Data: <searchLink fieldCode="AU" term="%22Gorman+DM%22">Gorman DM</searchLink>; School of Biomedical Sciences, The University of Queensland, Brisbane, Queensland 4072, Australia.<br /><searchLink fieldCode="AU" term="%22Li+XX%22">Li XX</searchLink>; School of Biomedical Sciences, The University of Queensland, Brisbane, Queensland 4072, Australia.<br /><searchLink fieldCode="AU" term="%22Lee+JD%22">Lee JD</searchLink>; School of Biomedical Sciences, The University of Queensland, Brisbane, Queensland 4072, Australia.<br /><searchLink fieldCode="AU" term="%22Fung+JN%22">Fung JN</searchLink>; School of Biomedical Sciences, The University of Queensland, Brisbane, Queensland 4072, Australia.<br /><searchLink fieldCode="AU" term="%22Cui+CS%22">Cui CS</searchLink>; School of Biomedical Sciences, The University of Queensland, Brisbane, Queensland 4072, Australia.<br /><searchLink fieldCode="AU" term="%22Lee+HS%22">Lee HS</searchLink>; School of Biomedical Sciences, The University of Queensland, Brisbane, Queensland 4072, Australia.<br /><searchLink fieldCode="AU" term="%22Rolfe+BE%22">Rolfe BE</searchLink>; Australian Institute for Bioengineering and Nanotechnology, The University of Queensland, Brisbane, Queensland 4072, Australia.<br /><searchLink fieldCode="AU" term="%22Woodruff+TM%22">Woodruff TM</searchLink>; School of Biomedical Sciences, The University of Queensland, Brisbane, Queensland 4072, Australia.; Queensland Brain Institute, The University of Queensland, Brisbane, Queensland 4072, Australia.<br /><searchLink fieldCode="AU" term="%22Clark+RJ%22">Clark RJ</searchLink>; School of Biomedical Sciences, The University of Queensland, Brisbane, Queensland 4072, Australia.
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  Data: <searchLink fieldCode="JN" term="%229716531%22">Journal of medicinal chemistry</searchLink> [J Med Chem] 2021 Nov 25; Vol. 64 (22), pp. 16598-16608. <i>Date of Electronic Publication: </i>2021 Nov 11.
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22American+Chemical+Society%22">American Chemical Society </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>9716531 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1520-4804 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2200222623%22">00222623 </searchLink><i>NLM ISO Abbreviation: </i>J Med Chem <i>Subsets: </i>MEDLINE
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        Value: 10.1021/acs.jmedchem.1c01174
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        Text: English
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              Text: 2021 Nov 25
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