Mechanistic Insights into a CDK9 Inhibitor Via Orthogonal Proteomics Methods.
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| Title: | Mechanistic Insights into a CDK9 Inhibitor Via Orthogonal Proteomics Methods. |
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| Authors: | Hendricks JA; Discovery Sciences, AstraZeneca, Boston, Massachusetts 02451, United States., Beaton N; Biognosys AG, Wagistrasse 21, Schlieren 8952, Switzerland., Chernobrovkin A; Pelago Bioscience AB, Banvaktsvägen 20, Solna 17148, Sweden., Miele E; Discovery Sciences, AstraZeneca, Boston, Massachusetts 02451, United States., Hamza GM; Discovery Sciences, AstraZeneca, Boston, Massachusetts 02451, United States.; Molecular, Cellular and Biomedical Sciences, University of New Hampshire, Durham, New Hampshire 03824, United States., Ricchiuto P; Discovery Sciences, AstraZeneca, Cambridge CB4 0WG, U.K., Tomlinson RC; Discovery Sciences, AstraZeneca, Boston, Massachusetts 02451, United States., Friman T; Pelago Bioscience AB, Banvaktsvägen 20, Solna 17148, Sweden., Borenstain C; Discovery Sciences, AstraZeneca, Boston, Massachusetts 02451, United States., Barlaam B; Oncology R&D, AstraZeneca, Cambridge CB4 0WG, U.K., Hande S; Oncology R&D, Boston, Massachusetts 02451, United States., Lamb ML; Oncology R&D, Boston, Massachusetts 02451, United States., De Savi C; Oncology R&D, Boston, Massachusetts 02451, United States., Davies R; Discovery Sciences, AstraZeneca, Cambridge CB4 0WG, U.K., Main M; Discovery Sciences, AstraZeneca, Cambridge CB4 0WG, U.K., Hellner J; Pelago Bioscience AB, Banvaktsvägen 20, Solna 17148, Sweden., Beeler K; Biognosys AG, Wagistrasse 21, Schlieren 8952, Switzerland., Feng Y; Biognosys AG, Wagistrasse 21, Schlieren 8952, Switzerland., Bruderer R; Biognosys AG, Wagistrasse 21, Schlieren 8952, Switzerland., Reiter L; Biognosys AG, Wagistrasse 21, Schlieren 8952, Switzerland., Molina DM; Pelago Bioscience AB, Banvaktsvägen 20, Solna 17148, Sweden., Castaldi MP; Discovery Sciences, AstraZeneca, Boston, Massachusetts 02451, United States. |
| Source: | ACS chemical biology [ACS Chem Biol] 2022 Jan 21; Vol. 17 (1), pp. 54-67. Date of Electronic Publication: 2021 Dec 25. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: American Chemical Society Country of Publication: United States NLM ID: 101282906 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1554-8937 (Electronic) Linking ISSN: 15548929 NLM ISO Abbreviation: ACS Chem Biol Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
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