A simple quinoline salt derivative is active in vitro against Plasmodiumfalciparum asexual blood stages and inhibits the development of cerebral malaria in murine model.

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Title: A simple quinoline salt derivative is active in vitro against Plasmodiumfalciparum asexual blood stages and inhibits the development of cerebral malaria in murine model.
Authors: Bezerra Bellei JC; Research Center Parasitology. Departament of Parasitology, Microbiology and Immunology. Federal University of Juiz de Fora, Juiz de Fora/MG 36.036-900, Brazil., Glanzmann N; Department of Chemistry, Institute of Exact Sciences, Federal University of Juiz de Fora, Juiz de Fora/MG 36.036-900, Brazil., Carpinter BA; Research Center Parasitology. Departament of Parasitology, Microbiology and Immunology. Federal University of Juiz de Fora, Juiz de Fora/MG 36.036-900, Brazil., Renhe DC; Research Center Parasitology. Departament of Parasitology, Microbiology and Immunology. Federal University of Juiz de Fora, Juiz de Fora/MG 36.036-900, Brazil., Marques CB; Research Center Parasitology. Departament of Parasitology, Microbiology and Immunology. Federal University of Juiz de Fora, Juiz de Fora/MG 36.036-900, Brazil., Azevedo MR; Research Center Parasitology. Departament of Parasitology, Microbiology and Immunology. Federal University of Juiz de Fora, Juiz de Fora/MG 36.036-900, Brazil., Barreto LM; Research Center Parasitology. Departament of Parasitology, Microbiology and Immunology. Federal University of Juiz de Fora, Juiz de Fora/MG 36.036-900, Brazil., Rocha VN; Research Center of Pathology and Veterinary Histology. Departament of Veterinary Medicine /Federal University of Juiz de Fora, Juiz de Fora/MG 36.036-900, Brazil., Karine da Costa Nunes I; Technological Development Support Laboratory, Chemistry Hub, Federal University of Rio de Janeiro, Rio de Janeiro/RJ 21.941-598, Brazil., Gualberto Pereira HM; Technological Development Support Laboratory, Chemistry Hub, Federal University of Rio de Janeiro, Rio de Janeiro/RJ 21.941-598, Brazil., Coimbra ES; Research Center Parasitology. Departament of Parasitology, Microbiology and Immunology. Federal University of Juiz de Fora, Juiz de Fora/MG 36.036-900, Brazil., Ferraz Coelho EA; Postgraduation Program in Health Sciences, Infectology and Tropical Medicine, Faculty of Medicine, Federal University of Minas Gerais, Av. Alfredo Balena, 190, 30130-100, Belo Horizonte, Minas Gerais, Brazil., David da Silva A; Department of Chemistry, Institute of Exact Sciences, Federal University of Juiz de Fora, Juiz de Fora/MG 36.036-900, Brazil., de Pilla Varotti F; Research Center on Biological Chemistry (NQBio)/Federal University of São João Del Rei, Divinópolis, MG, Brazil. Electronic address: varotti@ufsj.edu.br., Gorza Scopel KK; Research Center Parasitology. Departament of Parasitology, Microbiology and Immunology. Federal University of Juiz de Fora, Juiz de Fora/MG 36.036-900, Brazil. Electronic address: keziagscopel@gmail.com.
Source: Chemico-biological interactions [Chem Biol Interact] 2022 Mar 01; Vol. 355, pp. 109848. Date of Electronic Publication: 2022 Feb 09.
Publication Type: Journal Article
Journal Info: Publisher: Elsevier Country of Publication: Ireland NLM ID: 0227276 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1872-7786 (Electronic) Linking ISSN: 00092797 NLM ISO Abbreviation: Chem Biol Interact Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: A simple quinoline salt derivative is active in vitro against Plasmodiumfalciparum asexual blood stages and inhibits the development of cerebral malaria in murine model.
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  Data: <searchLink fieldCode="AU" term="%22Bezerra+Bellei+JC%22">Bezerra Bellei JC</searchLink>; Research Center Parasitology. Departament of Parasitology, Microbiology and Immunology. Federal University of Juiz de Fora, Juiz de Fora/MG 36.036-900, Brazil.<br /><searchLink fieldCode="AU" term="%22Glanzmann+N%22">Glanzmann N</searchLink>; Department of Chemistry, Institute of Exact Sciences, Federal University of Juiz de Fora, Juiz de Fora/MG 36.036-900, Brazil.<br /><searchLink fieldCode="AU" term="%22Carpinter+BA%22">Carpinter BA</searchLink>; Research Center Parasitology. Departament of Parasitology, Microbiology and Immunology. Federal University of Juiz de Fora, Juiz de Fora/MG 36.036-900, Brazil.<br /><searchLink fieldCode="AU" term="%22Renhe+DC%22">Renhe DC</searchLink>; Research Center Parasitology. Departament of Parasitology, Microbiology and Immunology. Federal University of Juiz de Fora, Juiz de Fora/MG 36.036-900, Brazil.<br /><searchLink fieldCode="AU" term="%22Marques+CB%22">Marques CB</searchLink>; Research Center Parasitology. Departament of Parasitology, Microbiology and Immunology. Federal University of Juiz de Fora, Juiz de Fora/MG 36.036-900, Brazil.<br /><searchLink fieldCode="AU" term="%22Azevedo+MR%22">Azevedo MR</searchLink>; Research Center Parasitology. Departament of Parasitology, Microbiology and Immunology. Federal University of Juiz de Fora, Juiz de Fora/MG 36.036-900, Brazil.<br /><searchLink fieldCode="AU" term="%22Barreto+LM%22">Barreto LM</searchLink>; Research Center Parasitology. Departament of Parasitology, Microbiology and Immunology. Federal University of Juiz de Fora, Juiz de Fora/MG 36.036-900, Brazil.<br /><searchLink fieldCode="AU" term="%22Rocha+VN%22">Rocha VN</searchLink>; Research Center of Pathology and Veterinary Histology. Departament of Veterinary Medicine /Federal University of Juiz de Fora, Juiz de Fora/MG 36.036-900, Brazil.<br /><searchLink fieldCode="AU" term="%22Karine+da+Costa+Nunes+I%22">Karine da Costa Nunes I</searchLink>; Technological Development Support Laboratory, Chemistry Hub, Federal University of Rio de Janeiro, Rio de Janeiro/RJ 21.941-598, Brazil.<br /><searchLink fieldCode="AU" term="%22Gualberto+Pereira+HM%22">Gualberto Pereira HM</searchLink>; Technological Development Support Laboratory, Chemistry Hub, Federal University of Rio de Janeiro, Rio de Janeiro/RJ 21.941-598, Brazil.<br /><searchLink fieldCode="AU" term="%22Coimbra+ES%22">Coimbra ES</searchLink>; Research Center Parasitology. Departament of Parasitology, Microbiology and Immunology. Federal University of Juiz de Fora, Juiz de Fora/MG 36.036-900, Brazil.<br /><searchLink fieldCode="AU" term="%22Ferraz+Coelho+EA%22">Ferraz Coelho EA</searchLink>; Postgraduation Program in Health Sciences, Infectology and Tropical Medicine, Faculty of Medicine, Federal University of Minas Gerais, Av. Alfredo Balena, 190, 30130-100, Belo Horizonte, Minas Gerais, Brazil.<br /><searchLink fieldCode="AU" term="%22David+da+Silva+A%22">David da Silva A</searchLink>; Department of Chemistry, Institute of Exact Sciences, Federal University of Juiz de Fora, Juiz de Fora/MG 36.036-900, Brazil.<br /><searchLink fieldCode="AU" term="%22de+Pilla+Varotti+F%22">de Pilla Varotti F</searchLink>; Research Center on Biological Chemistry (NQBio)/Federal University of São João Del Rei, Divinópolis, MG, Brazil. Electronic address: varotti@ufsj.edu.br.<br /><searchLink fieldCode="AU" term="%22Gorza+Scopel+KK%22">Gorza Scopel KK</searchLink>; Research Center Parasitology. Departament of Parasitology, Microbiology and Immunology. Federal University of Juiz de Fora, Juiz de Fora/MG 36.036-900, Brazil. Electronic address: keziagscopel@gmail.com.
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  Data: <searchLink fieldCode="JN" term="%220227276%22">Chemico-biological interactions</searchLink> [Chem Biol Interact] 2022 Mar 01; Vol. 355, pp. 109848. <i>Date of Electronic Publication: </i>2022 Feb 09.
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