CLIPSing Melanotan-II to Discover Multiple Functionally Selective hMCR Agonists.

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Bibliographic Details
Title: CLIPSing Melanotan-II to Discover Multiple Functionally Selective hMCR Agonists.
Authors: Tomassi S; Dipartimento di Farmacia, Università degli Studi di Napoli 'Federico II', Via D. Montesano 49, Naples 80131, Italy., Dimmito MP; Dipartimento di Farmacia, Università di Chieti-Pescara 'G. d'Annunzio', Via dei Vestini 31, Chieti 66100, Italy., Cai M; Department of Chemistry and Biochemistry, University of Arizona, Tucson, Arizona 85721, United States., D'Aniello A; DiSTABiF, University of Campania 'Luigi Vanvitelli', Via Vivaldi 43, 81100 Caserta, Italy., Del Bene A; DiSTABiF, University of Campania 'Luigi Vanvitelli', Via Vivaldi 43, 81100 Caserta, Italy., Messere A; DiSTABiF, University of Campania 'Luigi Vanvitelli', Via Vivaldi 43, 81100 Caserta, Italy., Liu Z; Department of Chemistry and Biochemistry, University of Arizona, Tucson, Arizona 85721, United States., Zhu T; Department of Chemistry and Biochemistry, University of Arizona, Tucson, Arizona 85721, United States., Hruby VJ; Department of Chemistry and Biochemistry, University of Arizona, Tucson, Arizona 85721, United States., Stefanucci A; Dipartimento di Farmacia, Università di Chieti-Pescara 'G. d'Annunzio', Via dei Vestini 31, Chieti 66100, Italy., Cosconati S; DiSTABiF, University of Campania 'Luigi Vanvitelli', Via Vivaldi 43, 81100 Caserta, Italy., Mollica A; Dipartimento di Farmacia, Università di Chieti-Pescara 'G. d'Annunzio', Via dei Vestini 31, Chieti 66100, Italy., Di Maro S; DiSTABiF, University of Campania 'Luigi Vanvitelli', Via Vivaldi 43, 81100 Caserta, Italy.
Source: Journal of medicinal chemistry [J Med Chem] 2022 Mar 10; Vol. 65 (5), pp. 4007-4017. Date of Electronic Publication: 2022 Feb 21.
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1520-4804
DOI:10.1021/acs.jmedchem.1c01848