New thiazole-based derivatives as EGFR/HER2 and DHFR inhibitors: Synthesis, molecular modeling simulations and anticancer activity.
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| Title: | New thiazole-based derivatives as EGFR/HER2 and DHFR inhibitors: Synthesis, molecular modeling simulations and anticancer activity. |
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| Authors: | Sabry MA; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, P.O. Box 35516, Mansoura, Egypt. Electronic address: mohamedamir@mans.edu.eg., Ghaly MA; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, P.O. Box 35516, Mansoura, Egypt. Electronic address: mariamaghaly@mans.edu.eg., Maarouf AR; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, P.O. Box 35516, Mansoura, Egypt., El-Subbagh HI; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, P.O. Box 35516, Mansoura, Egypt. Electronic address: subbagh@mans.edu.eg. |
| Source: | European journal of medicinal chemistry [Eur J Med Chem] 2022 Nov 05; Vol. 241, pp. 114661. Date of Electronic Publication: 2022 Aug 10. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1768-3254 (Electronic) Linking ISSN: 02235234 NLM ISO Abbreviation: Eur J Med Chem Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 35964425 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: New thiazole-based derivatives as EGFR/HER2 and DHFR inhibitors: Synthesis, molecular modeling simulations and anticancer activity. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Sabry+MA%22">Sabry MA</searchLink>; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, P.O. Box 35516, Mansoura, Egypt. Electronic address: mohamedamir@mans.edu.eg.<br /><searchLink fieldCode="AU" term="%22Ghaly+MA%22">Ghaly MA</searchLink>; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, P.O. Box 35516, Mansoura, Egypt. Electronic address: mariamaghaly@mans.edu.eg.<br /><searchLink fieldCode="AU" term="%22Maarouf+AR%22">Maarouf AR</searchLink>; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, P.O. Box 35516, Mansoura, Egypt.<br /><searchLink fieldCode="AU" term="%22El-Subbagh+HI%22">El-Subbagh HI</searchLink>; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, P.O. Box 35516, Mansoura, Egypt. Electronic address: subbagh@mans.edu.eg. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%220420510%22">European journal of medicinal chemistry</searchLink> [Eur J Med Chem] 2022 Nov 05; Vol. 241, pp. 114661. <i>Date of Electronic Publication: </i>2022 Aug 10. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Editions+Scientifiques+Elsevier%22">Editions Scientifiques Elsevier </searchLink><i>Country of Publication: </i>France <i>NLM ID: </i>0420510 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1768-3254 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2202235234%22">02235234 </searchLink><i>NLM ISO Abbreviation: </i>Eur J Med Chem <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=35964425 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1016/j.ejmech.2022.114661 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 114661 Titles: – TitleFull: New thiazole-based derivatives as EGFR/HER2 and DHFR inhibitors: Synthesis, molecular modeling simulations and anticancer activity. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Sabry MA – PersonEntity: Name: NameFull: Ghaly MA – PersonEntity: Name: NameFull: Maarouf AR – PersonEntity: Name: NameFull: El-Subbagh HI IsPartOfRelationships: – BibEntity: Dates: – D: 05 M: 11 Text: 2022 Nov 05 Type: published Y: 2022 Identifiers: – Type: issn-electronic Value: 1768-3254 Numbering: – Type: volume Value: 241 Titles: – TitleFull: European journal of medicinal chemistry Type: main |
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