Native Mass Spectrometry-Guided Screening Identifies Hit Fragments for HOP-HSP90 PPI Inhibition.

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Title: Native Mass Spectrometry-Guided Screening Identifies Hit Fragments for HOP-HSP90 PPI Inhibition.
Authors: Vaaltyn MC; The Biomedical Biotechnology Research Unit (BioBRU) Department of Biochemistry and Microbiology Department, Rhodes University, Makhanda, 6139, South Africa., Mateos-Jimenez M; EaStCHEM School of Chemistry, Joseph Black Building, David Brewster Road, Edinburgh, EH93FJ, UK., Müller R; School of Chemistry and Physics, University of KwaZulu-Natal, Scottsville, 3209, South Africa., Mackay CL; EaStCHEM School of Chemistry, Joseph Black Building, David Brewster Road, Edinburgh, EH93FJ, UK., Edkins AL; The Biomedical Biotechnology Research Unit (BioBRU) Department of Biochemistry and Microbiology Department, Rhodes University, Makhanda, 6139, South Africa., Clarke DJ; EaStCHEM School of Chemistry, Joseph Black Building, David Brewster Road, Edinburgh, EH93FJ, UK., Veale CGL; Department of Chemistry, University of Cape Town Rondebosch, Cape Town, 7700, South Africa.
Source: Chembiochem : a European journal of chemical biology [Chembiochem] 2022 Nov 04; Vol. 23 (21), pp. e202200322. Date of Electronic Publication: 2022 Sep 20.
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
Journal Info: Publisher: Wiley-VCH Verlag Country of Publication: Germany NLM ID: 100937360 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1439-7633 (Electronic) Linking ISSN: 14394227 NLM ISO Abbreviation: Chembiochem Subsets: MEDLINE
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  Data: Native Mass Spectrometry-Guided Screening Identifies Hit Fragments for HOP-HSP90 PPI Inhibition.
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  Data: <searchLink fieldCode="AU" term="%22Vaaltyn+MC%22">Vaaltyn MC</searchLink>; The Biomedical Biotechnology Research Unit (BioBRU) Department of Biochemistry and Microbiology Department, Rhodes University, Makhanda, 6139, South Africa.<br /><searchLink fieldCode="AU" term="%22Mateos-Jimenez+M%22">Mateos-Jimenez M</searchLink>; EaStCHEM School of Chemistry, Joseph Black Building, David Brewster Road, Edinburgh, EH93FJ, UK.<br /><searchLink fieldCode="AU" term="%22Müller+R%22">Müller R</searchLink>; School of Chemistry and Physics, University of KwaZulu-Natal, Scottsville, 3209, South Africa.<br /><searchLink fieldCode="AU" term="%22Mackay+CL%22">Mackay CL</searchLink>; EaStCHEM School of Chemistry, Joseph Black Building, David Brewster Road, Edinburgh, EH93FJ, UK.<br /><searchLink fieldCode="AU" term="%22Edkins+AL%22">Edkins AL</searchLink>; The Biomedical Biotechnology Research Unit (BioBRU) Department of Biochemistry and Microbiology Department, Rhodes University, Makhanda, 6139, South Africa.<br /><searchLink fieldCode="AU" term="%22Clarke+DJ%22">Clarke DJ</searchLink>; EaStCHEM School of Chemistry, Joseph Black Building, David Brewster Road, Edinburgh, EH93FJ, UK.<br /><searchLink fieldCode="AU" term="%22Veale+CGL%22">Veale CGL</searchLink>; Department of Chemistry, University of Cape Town Rondebosch, Cape Town, 7700, South Africa.
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  Data: <searchLink fieldCode="JN" term="%22100937360%22">Chembiochem : a European journal of chemical biology</searchLink> [Chembiochem] 2022 Nov 04; Vol. 23 (21), pp. e202200322. <i>Date of Electronic Publication: </i>2022 Sep 20.
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Wiley-VCH+Verlag%22">Wiley-VCH Verlag </searchLink><i>Country of Publication: </i>Germany <i>NLM ID: </i>100937360 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1439-7633 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2214394227%22">14394227 </searchLink><i>NLM ISO Abbreviation: </i>Chembiochem <i>Subsets: </i>MEDLINE
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        Value: 10.1002/cbic.202200322
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      – TitleFull: Native Mass Spectrometry-Guided Screening Identifies Hit Fragments for HOP-HSP90 PPI Inhibition.
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              Text: 2022 Nov 04
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