Native Mass Spectrometry-Guided Screening Identifies Hit Fragments for HOP-HSP90 PPI Inhibition.
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| Title: | Native Mass Spectrometry-Guided Screening Identifies Hit Fragments for HOP-HSP90 PPI Inhibition. |
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| Authors: | Vaaltyn MC; The Biomedical Biotechnology Research Unit (BioBRU) Department of Biochemistry and Microbiology Department, Rhodes University, Makhanda, 6139, South Africa., Mateos-Jimenez M; EaStCHEM School of Chemistry, Joseph Black Building, David Brewster Road, Edinburgh, EH93FJ, UK., Müller R; School of Chemistry and Physics, University of KwaZulu-Natal, Scottsville, 3209, South Africa., Mackay CL; EaStCHEM School of Chemistry, Joseph Black Building, David Brewster Road, Edinburgh, EH93FJ, UK., Edkins AL; The Biomedical Biotechnology Research Unit (BioBRU) Department of Biochemistry and Microbiology Department, Rhodes University, Makhanda, 6139, South Africa., Clarke DJ; EaStCHEM School of Chemistry, Joseph Black Building, David Brewster Road, Edinburgh, EH93FJ, UK., Veale CGL; Department of Chemistry, University of Cape Town Rondebosch, Cape Town, 7700, South Africa. |
| Source: | Chembiochem : a European journal of chemical biology [Chembiochem] 2022 Nov 04; Vol. 23 (21), pp. e202200322. Date of Electronic Publication: 2022 Sep 20. |
| Publication Type: | Journal Article; Research Support, Non-U.S. Gov't |
| Journal Info: | Publisher: Wiley-VCH Verlag Country of Publication: Germany NLM ID: 100937360 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1439-7633 (Electronic) Linking ISSN: 14394227 NLM ISO Abbreviation: Chembiochem Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 36017658 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Native Mass Spectrometry-Guided Screening Identifies Hit Fragments for HOP-HSP90 PPI Inhibition. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Vaaltyn+MC%22">Vaaltyn MC</searchLink>; The Biomedical Biotechnology Research Unit (BioBRU) Department of Biochemistry and Microbiology Department, Rhodes University, Makhanda, 6139, South Africa.<br /><searchLink fieldCode="AU" term="%22Mateos-Jimenez+M%22">Mateos-Jimenez M</searchLink>; EaStCHEM School of Chemistry, Joseph Black Building, David Brewster Road, Edinburgh, EH93FJ, UK.<br /><searchLink fieldCode="AU" term="%22Müller+R%22">Müller R</searchLink>; School of Chemistry and Physics, University of KwaZulu-Natal, Scottsville, 3209, South Africa.<br /><searchLink fieldCode="AU" term="%22Mackay+CL%22">Mackay CL</searchLink>; EaStCHEM School of Chemistry, Joseph Black Building, David Brewster Road, Edinburgh, EH93FJ, UK.<br /><searchLink fieldCode="AU" term="%22Edkins+AL%22">Edkins AL</searchLink>; The Biomedical Biotechnology Research Unit (BioBRU) Department of Biochemistry and Microbiology Department, Rhodes University, Makhanda, 6139, South Africa.<br /><searchLink fieldCode="AU" term="%22Clarke+DJ%22">Clarke DJ</searchLink>; EaStCHEM School of Chemistry, Joseph Black Building, David Brewster Road, Edinburgh, EH93FJ, UK.<br /><searchLink fieldCode="AU" term="%22Veale+CGL%22">Veale CGL</searchLink>; Department of Chemistry, University of Cape Town Rondebosch, Cape Town, 7700, South Africa. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%22100937360%22">Chembiochem : a European journal of chemical biology</searchLink> [Chembiochem] 2022 Nov 04; Vol. 23 (21), pp. e202200322. <i>Date of Electronic Publication: </i>2022 Sep 20. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article; Research Support, Non-U.S. Gov't – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Wiley-VCH+Verlag%22">Wiley-VCH Verlag </searchLink><i>Country of Publication: </i>Germany <i>NLM ID: </i>100937360 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1439-7633 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2214394227%22">14394227 </searchLink><i>NLM ISO Abbreviation: </i>Chembiochem <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=36017658 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1002/cbic.202200322 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: e202200322 Titles: – TitleFull: Native Mass Spectrometry-Guided Screening Identifies Hit Fragments for HOP-HSP90 PPI Inhibition. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Vaaltyn MC – PersonEntity: Name: NameFull: Mateos-Jimenez M – PersonEntity: Name: NameFull: Müller R – PersonEntity: Name: NameFull: Mackay CL – PersonEntity: Name: NameFull: Edkins AL – PersonEntity: Name: NameFull: Clarke DJ – PersonEntity: Name: NameFull: Veale CGL IsPartOfRelationships: – BibEntity: Dates: – D: 04 M: 11 Text: 2022 Nov 04 Type: published Y: 2022 Identifiers: – Type: issn-electronic Value: 1439-7633 Numbering: – Type: volume Value: 23 – Type: issue Value: 21 Titles: – TitleFull: Chembiochem : a European journal of chemical biology Type: main |
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