Evaluation of the histamine H3 receptor antagonists from LINS01 series as cholinesterases inhibitors: Enzymatic and modeling studies.

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Title: Evaluation of the histamine H3 receptor antagonists from LINS01 series as cholinesterases inhibitors: Enzymatic and modeling studies.
Authors: Lopes FB; Department of Pharmaceutical Sciences, Universidade Federal de São Paulo (Unifesp), Diadema, Brazil., Aranha CMSQ; Department of Pharmaceutical Sciences, Universidade Federal de São Paulo (Unifesp), Diadema, Brazil., Corrêa MF; Department of Medicine, Universidade Federal de São Paulo (Unifesp), São Paulo, Brazil., Fernandes GAB; Department of Pharmaceutical Sciences, Universidade Federal de São Paulo (Unifesp), Diadema, Brazil., Okamoto DN; Department of Pharmaceutical Sciences, Universidade Federal de São Paulo (Unifesp), Diadema, Brazil., Simões LPM; Department of Biochemistry and Organic Chemistry, Institute of Chemistry, São Paulo State University (Unesp), Araraquara, Brazil., Junior NMN; Department of Biochemistry and Organic Chemistry, Institute of Chemistry, São Paulo State University (Unesp), Araraquara, Brazil., Fernandes JPS; Department of Pharmaceutical Sciences, Universidade Federal de São Paulo (Unifesp), Diadema, Brazil.
Source: Chemical biology & drug design [Chem Biol Drug Des] 2022 Nov; Vol. 100 (5), pp. 722-729. Date of Electronic Publication: 2022 Sep 08.
Publication Type: Letter; Research Support, Non-U.S. Gov't
Journal Info: Publisher: Wiley-Blackwell Country of Publication: England NLM ID: 101262549 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1747-0285 (Electronic) Linking ISSN: 17470277 NLM ISO Abbreviation: Chem Biol Drug Des Subsets: MEDLINE
Database: MEDLINE Ultimate
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ISSN:1747-0285
DOI:10.1111/cbdd.14139