Opportunities and challenges for the development of M1 muscarinic receptor positive allosteric modulators in the treatment for neurocognitive deficits.

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Title: Opportunities and challenges for the development of M1 muscarinic receptor positive allosteric modulators in the treatment for neurocognitive deficits.
Authors: Nguyen HTM; Drug Discovery Biology, Monash University, Parkville, Melbourne, VIC, Australia.; Department of Biochemistry, Hanoi University of Pharmacy, Hanoi, Vietnam., van der Westhuizen ET; Drug Discovery Biology, Monash University, Parkville, Melbourne, VIC, Australia., Langmead CJ; Drug Discovery Biology, Monash University, Parkville, Melbourne, VIC, Australia.; Neuromedicines Discovery Centre, Monash University, Parkville, Melbourne, VIC, Australia.; ARC Centre for Cryo-electron Microscopy of Membrane Proteins, Monash University, Parkville, Melbourne, VIC, Australia., Tobin AB; Centre for Translational Pharmacology, University of Glasgow, Glasgow, UK., Sexton PM; Drug Discovery Biology, Monash University, Parkville, Melbourne, VIC, Australia.; ARC Centre for Cryo-electron Microscopy of Membrane Proteins, Monash University, Parkville, Melbourne, VIC, Australia., Christopoulos A; Drug Discovery Biology, Monash University, Parkville, Melbourne, VIC, Australia.; Neuromedicines Discovery Centre, Monash University, Parkville, Melbourne, VIC, Australia.; ARC Centre for Cryo-electron Microscopy of Membrane Proteins, Monash University, Parkville, Melbourne, VIC, Australia., Valant C; Drug Discovery Biology, Monash University, Parkville, Melbourne, VIC, Australia.; Neuromedicines Discovery Centre, Monash University, Parkville, Melbourne, VIC, Australia.
Source: British journal of pharmacology [Br J Pharmacol] 2024 Jul; Vol. 181 (14), pp. 2114-2142. Date of Electronic Publication: 2022 Dec 04.
Publication Type: Journal Article; Review
Journal Info: Publisher: Wiley Country of Publication: England NLM ID: 7502536 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1476-5381 (Electronic) Linking ISSN: 00071188 NLM ISO Abbreviation: Br J Pharmacol Subsets: MEDLINE
Database: MEDLINE Ultimate
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ISSN:1476-5381
DOI:10.1111/bph.15982