Discovery of High-Affinity Small-Molecule Binders of the Epigenetic Reader YEATS4.

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Bibliographic Details
Title: Discovery of High-Affinity Small-Molecule Binders of the Epigenetic Reader YEATS4.
Authors: Londregan AT; Pfizer Medicine Design, Pfizer Worldwide Research and Development, Cambridge, Massachusetts 02139, United States., Aitmakhanova K; Centre for Medicines Discovery, NDM, University of Oxford, Oxford OX3 7DQ, U.K., Bennett J; Centre for Medicines Discovery, NDM, University of Oxford, Oxford OX3 7DQ, U.K., Byrnes LJ; Pfizer Worldwide Research and Development, Groton, Connecticut 06340, United States., Canterbury DP; Pfizer Worldwide Research and Development, Groton, Connecticut 06340, United States., Cheng X; Pfizer Worldwide Research and Development, Cambridge, Massachusetts 02139, United States., Christott T; Centre for Medicines Discovery, NDM, University of Oxford, Oxford OX3 7DQ, U.K., Clemens J; Pfizer Worldwide Research and Development, Groton, Connecticut 06340, United States., Coffey SB; Pfizer Worldwide Research and Development, Groton, Connecticut 06340, United States., Dias JM; Pfizer Worldwide Research and Development, Groton, Connecticut 06340, United States., Dowling MS; Pfizer Worldwide Research and Development, Groton, Connecticut 06340, United States., Farnie G; Centre for Medicines Discovery, NDM, University of Oxford, Oxford OX3 7DQ, U.K., Fedorov O; Centre for Medicines Discovery, NDM, University of Oxford, Oxford OX3 7DQ, U.K., Fennell KF; Pfizer Worldwide Research and Development, Groton, Connecticut 06340, United States., Gamble V; Centre for Medicines Discovery, NDM, University of Oxford, Oxford OX3 7DQ, U.K., Gileadi C; Centre for Medicines Discovery, NDM, University of Oxford, Oxford OX3 7DQ, U.K., Giroud C; Centre for Medicines Discovery, NDM, University of Oxford, Oxford OX3 7DQ, U.K., Harris MR; Pfizer Worldwide Research and Development, Groton, Connecticut 06340, United States., Hollingshead BD; Pfizer Worldwide Research and Development, Cambridge, Massachusetts 02139, United States., Huber K; Centre for Medicines Discovery, NDM, University of Oxford, Oxford OX3 7DQ, U.K., Korczynska M; Pfizer Worldwide Research and Development, Cambridge, Massachusetts 02139, United States., Lapham K; Pfizer Worldwide Research and Development, Groton, Connecticut 06340, United States., Loria PM; Pfizer Worldwide Research and Development, Groton, Connecticut 06340, United States., Narayanan A; Pfizer Worldwide Research and Development, Cambridge, Massachusetts 02139, United States., Owen DR; Pfizer Worldwide Research and Development, Cambridge, Massachusetts 02139, United States., Raux B; Centre for Medicines Discovery, NDM, University of Oxford, Oxford OX3 7DQ, U.K., Sahasrabudhe PV; Pfizer Worldwide Research and Development, Groton, Connecticut 06340, United States., Ruggeri RB; Pfizer Worldwide Research and Development, Groton, Connecticut 06340, United States., Sáez LD; Centre for Medicines Discovery, NDM, University of Oxford, Oxford OX3 7DQ, U.K., Stock IA; Pfizer Worldwide Research and Development, Groton, Connecticut 06340, United States., Thuma BA; Pfizer Worldwide Research and Development, Groton, Connecticut 06340, United States., Tsai A; Pfizer Worldwide Research and Development, Groton, Connecticut 06340, United States., Varghese AE; Pfizer Worldwide Research and Development, Groton, Connecticut 06340, United States.
Source: Journal of medicinal chemistry [J Med Chem] 2023 Jan 12; Vol. 66 (1), pp. 460-472. Date of Electronic Publication: 2022 Dec 23.
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1520-4804
DOI:10.1021/acs.jmedchem.2c01421