Discovery of Selective Tertiary Amide Inhibitors of Cyclin-Dependent Kinase 2 (CDK2).

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Bibliographic Details
Title: Discovery of Selective Tertiary Amide Inhibitors of Cyclin-Dependent Kinase 2 (CDK2).
Authors: Zeng M; Genentech Inc., South San Francisco, California 94080, United States., Grandner JM; Genentech Inc., South San Francisco, California 94080, United States., Bryan MC; Janssen R&D, 1400 McKean Rd, Spring House, Pennsylvania 19002, United States., Verma V; Genentech Inc., South San Francisco, California 94080, United States., Larouche-Gauthier R; Paraza Pharma Inc., Montreal, QC H4S 2E1, Canada., Leclerc JP; Paraza Pharma Inc., Montreal, QC H4S 2E1, Canada., Zhao L; Paraza Pharma Inc., Montreal, QC H4S 2E1, Canada., Haghshenas P; Paraza Pharma Inc., Montreal, QC H4S 2E1, Canada., Aubert-Nicol S; Paraza Pharma Inc., Montreal, QC H4S 2E1, Canada., Yadav A; Paraza Pharma Inc., Montreal, QC H4S 2E1, Canada., Ashley M; Genentech Inc., South San Francisco, California 94080, United States., Chen JZ; Genentech Inc., South San Francisco, California 94080, United States., Durk M; Genentech Inc., South San Francisco, California 94080, United States., Samy KE; Genentech Inc., South San Francisco, California 94080, United States., Nespi M; Genentech Inc., South San Francisco, California 94080, United States., Levy E; Genentech Inc., South San Francisco, California 94080, United States., Merrick K; Genentech Inc., South San Francisco, California 94080, United States., Moffat JG; Genentech Inc., South San Francisco, California 94080, United States., Murray J; Genentech Inc., South San Francisco, California 94080, United States., Oh A; Genentech Inc., South San Francisco, California 94080, United States., Orr C; Genentech Inc., South San Francisco, California 94080, United States., Segal E; Genentech Inc., South San Francisco, California 94080, United States., Sims J; Genentech Inc., South San Francisco, California 94080, United States., Sneeringer C; Genentech Inc., South San Francisco, California 94080, United States., Prangley M; Genentech Inc., South San Francisco, California 94080, United States., Vartanian S; Genentech Inc., South San Francisco, California 94080, United States., Magnuson S; Genentech Inc., South San Francisco, California 94080, United States., Parr BT; Genentech Inc., South San Francisco, California 94080, United States.
Source: ACS medicinal chemistry letters [ACS Med Chem Lett] 2023 Aug 24; Vol. 14 (9), pp. 1179-1187. Date of Electronic Publication: 2023 Aug 24 (Print Publication: 2023).
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1948-5875
DOI:10.1021/acsmedchemlett.3c00142