Synthesis and structure-activity relationships of aryl fluorosulfate-based inhibitors as novel antitubercular agents.
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| Title: | Synthesis and structure-activity relationships of aryl fluorosulfate-based inhibitors as novel antitubercular agents. |
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| Authors: | Yang B; Calibr, a Division of Scripps Research, La Jolla, CA 92037, USA. Electronic address: byang@scripps.edu., Sukheja P; Calibr, a Division of Scripps Research, La Jolla, CA 92037, USA., Qin B; Calibr, a Division of Scripps Research, La Jolla, CA 92037, USA., Li G; Department of Chemistry, Scripps Research, La Jolla, CA 92037, USA., Bare GAL; Department of Chemistry, Scripps Research, La Jolla, CA 92037, USA., Cascioferro A; Calibr, a Division of Scripps Research, La Jolla, CA 92037, USA., Love MS; Calibr, a Division of Scripps Research, La Jolla, CA 92037, USA., Petrassi HM; Calibr, a Division of Scripps Research, La Jolla, CA 92037, USA., Sharpless KB; Department of Chemistry, Scripps Research, La Jolla, CA 92037, USA., McNamara CW; Calibr, a Division of Scripps Research, La Jolla, CA 92037, USA., Chatterjee AK; Calibr, a Division of Scripps Research, La Jolla, CA 92037, USA. |
| Source: | Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2024 Jan 15; Vol. 98, pp. 129596. Date of Electronic Publication: 2023 Dec 23. |
| Publication Type: | Journal Article; Research Support, Non-U.S. Gov't |
| Journal Info: | Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
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