Early pharmacological profiling of isatin derivatives as potent and selective cytotoxic agents.

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Title: Early pharmacological profiling of isatin derivatives as potent and selective cytotoxic agents.
Authors: Puerta A; BioLab, Instituto Universitario de Bio-Orgánica Antonio González (IUBO-AG), Universidad de La Laguna, PO Box 456, 38200 La Laguna, Spain., González-Bakker A; BioLab, Instituto Universitario de Bio-Orgánica Antonio González (IUBO-AG), Universidad de La Laguna, PO Box 456, 38200 La Laguna, Spain., Brandão P; Egas Moniz Center for Interdisciplinary Research (CiiEM), Egas Moniz School of Health & Science, 2829-511 Almada, Portugal; iBB-Institute for Bioengineering and Biosciences, Department of Bioengineering, and Associate Laboratory i4HB-Institute for Health and Bio-Economy, Instituto Superior Técnico, University of Lisboa, Av. Rovisco Pais, 1049-001 Lisbon, Portugal; Centro de Química de Coimbra - Institute of Molecular Sciences (CQC-IMS), Departamento de Química, Faculdade de Ciências e Tecnologia, University of Coimbra, 3004-535 Coimbra, Portugal., Pineiro M; Centro de Química de Coimbra - Institute of Molecular Sciences (CQC-IMS), Departamento de Química, Faculdade de Ciências e Tecnologia, University of Coimbra, 3004-535 Coimbra, Portugal., Burke AJ; Centro de Química de Coimbra - Institute of Molecular Sciences (CQC-IMS), Departamento de Química, Faculdade de Ciências e Tecnologia, University of Coimbra, 3004-535 Coimbra, Portugal; Faculty Pharmacy, University of Coimbra, Pólo das Ciências da Saúde, Azinhaga de Santa Comba, 3000-548 Coimbra, Portugal., Giovannetti E; Department of Medical Oncology, Cancer Center Amsterdam, Amsterdam University Medical Centers (Amsterdam UMC), Vrije Universiteit Amsterdam, The Netherlands; Cancer Pharmacology Lab, Fondazione Pisana per la Scienza, Pisa, Italy., Fernandes MX; Department of Engineering and Chemical Sciences, Karlstad University, 65188 Karlstad, Sweden., Padrón JM; BioLab, Instituto Universitario de Bio-Orgánica Antonio González (IUBO-AG), Universidad de La Laguna, PO Box 456, 38200 La Laguna, Spain. Electronic address: jmpadron@ull.es.
Source: Biochemical pharmacology [Biochem Pharmacol] 2024 Apr; Vol. 222, pp. 116059. Date of Electronic Publication: 2024 Feb 15.
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
Journal Info: Publisher: Elsevier Science Country of Publication: England NLM ID: 0101032 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1873-2968 (Electronic) Linking ISSN: 00062952 NLM ISO Abbreviation: Biochem Pharmacol Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1873-2968
DOI:10.1016/j.bcp.2024.116059