Enhancing the Small-Scale Screenable Biological Space beyond Known Chemogenomics Libraries with Gray Chemical Matter─Compounds with Novel Mechanisms from High-Throughput Screening Profiles.

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Title: Enhancing the Small-Scale Screenable Biological Space beyond Known Chemogenomics Libraries with Gray Chemical Matter─Compounds with Novel Mechanisms from High-Throughput Screening Profiles.
Authors: Thomas JR; Novartis Biomedical Research, Cambridge, Massachusetts 02139, United States., Shelton C 4th; Novartis Biomedical Research, Cambridge, Massachusetts 02139, United States., Murphy J; Novartis Biomedical Research, Cambridge, Massachusetts 02139, United States., Brittain S; Novartis Biomedical Research, Cambridge, Massachusetts 02139, United States., Bray MA; Novartis Biomedical Research, Cambridge, Massachusetts 02139, United States., Aspesi P; Novartis Biomedical Research, Cambridge, Massachusetts 02139, United States., Concannon J; Novartis Biomedical Research, Cambridge, Massachusetts 02139, United States., King FJ; Novartis Biomedical Research, San Diego, California 92121, United States., Ihry RJ; Novartis Biomedical Research, San Diego, California 92121, United States., Ho DJ; Novartis Biomedical Research, San Diego, California 92121, United States., Henault M; Novartis Biomedical Research, Cambridge, Massachusetts 02139, United States., Hadjikyriacou A; Novartis Biomedical Research, Cambridge, Massachusetts 02139, United States., Neri M; Novartis Biomedical Research, Basel 4056, Switzerland., Sigoillot FD; Novartis Biomedical Research, Cambridge, Massachusetts 02139, United States., Pham HT; Novartis Biomedical Research, Cambridge, Massachusetts 02139, United States., Shum M; Novartis Biomedical Research, Cambridge, Massachusetts 02139, United States., Barys L; Novartis Biomedical Research, Basel 4056, Switzerland., Jones MD; Novartis Biomedical Research, Cambridge, Massachusetts 02139, United States., Martin EJ; Novartis Biomedical Research, Emeryville, California 94608, United States., Blechschmidt A; Novartis Biomedical Research, Basel 4056, Switzerland., Rieffel S; Novartis Biomedical Research, Basel 4056, Switzerland., Troxler TJ; Novartis Biomedical Research, Basel 4056, Switzerland., Mapa FA; Novartis Biomedical Research, Cambridge, Massachusetts 02139, United States., Jenkins JL; Novartis Biomedical Research, Cambridge, Massachusetts 02139, United States., Jain RK; Novartis Biomedical Research, Cambridge, Massachusetts 02139, United States., Kutchukian PS; Novartis Biomedical Research, Cambridge, Massachusetts 02139, United States., Schirle M; Novartis Biomedical Research, Cambridge, Massachusetts 02139, United States., Renner S; Novartis Biomedical Research, Basel 4056, Switzerland.
Source: ACS chemical biology [ACS Chem Biol] 2024 Apr 19; Vol. 19 (4), pp. 938-952. Date of Electronic Publication: 2024 Apr 02.
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101282906 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1554-8937 (Electronic) Linking ISSN: 15548929 NLM ISO Abbreviation: ACS Chem Biol Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1554-8937
DOI:10.1021/acschembio.3c00737