Characterisation of high throughput screening outputs for small molecule degrader discovery.
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| Title: | Characterisation of high throughput screening outputs for small molecule degrader discovery. |
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| Authors: | Bell LE; Research Institute of Molecular Pathology (IMP), Vienna BioCenter (VBC), Campus-Vienna-BioCenter 1, 1030 Vienna, Austria; Vienna BioCenter PhD Program, Doctoral School of the University of Vienna and Medical University of Vienna, 1030, Vienna, Austria., Bardelle C; Hit Discovery, Discovery Sciences, R&D, AstraZeneca, Alderley Park, Macclesfield, UK., Packer MJ; TDE, Oncology, R&D, AstraZeneca, Cambridge, UK., Kastl J; Assay.Works GmbH, Am Biopark 11, Regensburg, Germany., Holdgate GA; Hit Discovery, Discovery Sciences, R&D, AstraZeneca, Alderley Park, Macclesfield, UK. Electronic address: geoff.holdgate@astrazeneca.com., Davies G; Hit Discovery, Discovery Sciences, R&D, AstraZeneca, Alderley Park, Macclesfield, UK. |
| Source: | SLAS discovery : advancing life sciences R & D [SLAS Discov] 2024 Jul; Vol. 29 (5), pp. 100162. Date of Electronic Publication: 2024 May 24. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: SAGE Publications Country of Publication: United States NLM ID: 101697563 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2472-5560 (Electronic) Linking ISSN: 24725552 NLM ISO Abbreviation: SLAS Discov Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 38797285 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Characterisation of high throughput screening outputs for small molecule degrader discovery. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Bell+LE%22">Bell LE</searchLink>; Research Institute of Molecular Pathology (IMP), Vienna BioCenter (VBC), Campus-Vienna-BioCenter 1, 1030 Vienna, Austria; Vienna BioCenter PhD Program, Doctoral School of the University of Vienna and Medical University of Vienna, 1030, Vienna, Austria.<br /><searchLink fieldCode="AU" term="%22Bardelle+C%22">Bardelle C</searchLink>; Hit Discovery, Discovery Sciences, R&D, AstraZeneca, Alderley Park, Macclesfield, UK.<br /><searchLink fieldCode="AU" term="%22Packer+MJ%22">Packer MJ</searchLink>; TDE, Oncology, R&D, AstraZeneca, Cambridge, UK.<br /><searchLink fieldCode="AU" term="%22Kastl+J%22">Kastl J</searchLink>; Assay.Works GmbH, Am Biopark 11, Regensburg, Germany.<br /><searchLink fieldCode="AU" term="%22Holdgate+GA%22">Holdgate GA</searchLink>; Hit Discovery, Discovery Sciences, R&D, AstraZeneca, Alderley Park, Macclesfield, UK. Electronic address: geoff.holdgate@astrazeneca.com.<br /><searchLink fieldCode="AU" term="%22Davies+G%22">Davies G</searchLink>; Hit Discovery, Discovery Sciences, R&D, AstraZeneca, Alderley Park, Macclesfield, UK. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%22101697563%22">SLAS discovery : advancing life sciences R & D</searchLink> [SLAS Discov] 2024 Jul; Vol. 29 (5), pp. 100162. <i>Date of Electronic Publication: </i>2024 May 24. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22SAGE+Publications%22">SAGE Publications </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>101697563 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>2472-5560 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2224725552%22">24725552 </searchLink><i>NLM ISO Abbreviation: </i>SLAS Discov <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=38797285 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1016/j.slasd.2024.100162 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 100162 Titles: – TitleFull: Characterisation of high throughput screening outputs for small molecule degrader discovery. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Bell LE – PersonEntity: Name: NameFull: Bardelle C – PersonEntity: Name: NameFull: Packer MJ – PersonEntity: Name: NameFull: Kastl J – PersonEntity: Name: NameFull: Holdgate GA – PersonEntity: Name: NameFull: Davies G IsPartOfRelationships: – BibEntity: Dates: – D: 01 M: 07 Text: 2024 Jul Type: published Y: 2024 Identifiers: – Type: issn-electronic Value: 2472-5560 Numbering: – Type: volume Value: 29 – Type: issue Value: 5 Titles: – TitleFull: SLAS discovery : advancing life sciences R & D Type: main |
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