Characterisation of high throughput screening outputs for small molecule degrader discovery.

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Title: Characterisation of high throughput screening outputs for small molecule degrader discovery.
Authors: Bell LE; Research Institute of Molecular Pathology (IMP), Vienna BioCenter (VBC), Campus-Vienna-BioCenter 1, 1030 Vienna, Austria; Vienna BioCenter PhD Program, Doctoral School of the University of Vienna and Medical University of Vienna, 1030, Vienna, Austria., Bardelle C; Hit Discovery, Discovery Sciences, R&D, AstraZeneca, Alderley Park, Macclesfield, UK., Packer MJ; TDE, Oncology, R&D, AstraZeneca, Cambridge, UK., Kastl J; Assay.Works GmbH, Am Biopark 11, Regensburg, Germany., Holdgate GA; Hit Discovery, Discovery Sciences, R&D, AstraZeneca, Alderley Park, Macclesfield, UK. Electronic address: geoff.holdgate@astrazeneca.com., Davies G; Hit Discovery, Discovery Sciences, R&D, AstraZeneca, Alderley Park, Macclesfield, UK.
Source: SLAS discovery : advancing life sciences R & D [SLAS Discov] 2024 Jul; Vol. 29 (5), pp. 100162. Date of Electronic Publication: 2024 May 24.
Publication Type: Journal Article
Journal Info: Publisher: SAGE Publications Country of Publication: United States NLM ID: 101697563 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2472-5560 (Electronic) Linking ISSN: 24725552 NLM ISO Abbreviation: SLAS Discov Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: Characterisation of high throughput screening outputs for small molecule degrader discovery.
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  Data: <searchLink fieldCode="AU" term="%22Bell+LE%22">Bell LE</searchLink>; Research Institute of Molecular Pathology (IMP), Vienna BioCenter (VBC), Campus-Vienna-BioCenter 1, 1030 Vienna, Austria; Vienna BioCenter PhD Program, Doctoral School of the University of Vienna and Medical University of Vienna, 1030, Vienna, Austria.<br /><searchLink fieldCode="AU" term="%22Bardelle+C%22">Bardelle C</searchLink>; Hit Discovery, Discovery Sciences, R&D, AstraZeneca, Alderley Park, Macclesfield, UK.<br /><searchLink fieldCode="AU" term="%22Packer+MJ%22">Packer MJ</searchLink>; TDE, Oncology, R&D, AstraZeneca, Cambridge, UK.<br /><searchLink fieldCode="AU" term="%22Kastl+J%22">Kastl J</searchLink>; Assay.Works GmbH, Am Biopark 11, Regensburg, Germany.<br /><searchLink fieldCode="AU" term="%22Holdgate+GA%22">Holdgate GA</searchLink>; Hit Discovery, Discovery Sciences, R&D, AstraZeneca, Alderley Park, Macclesfield, UK. Electronic address: geoff.holdgate@astrazeneca.com.<br /><searchLink fieldCode="AU" term="%22Davies+G%22">Davies G</searchLink>; Hit Discovery, Discovery Sciences, R&D, AstraZeneca, Alderley Park, Macclesfield, UK.
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  Data: <searchLink fieldCode="JN" term="%22101697563%22">SLAS discovery : advancing life sciences R & D</searchLink> [SLAS Discov] 2024 Jul; Vol. 29 (5), pp. 100162. <i>Date of Electronic Publication: </i>2024 May 24.
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22SAGE+Publications%22">SAGE Publications </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>101697563 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>2472-5560 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2224725552%22">24725552 </searchLink><i>NLM ISO Abbreviation: </i>SLAS Discov <i>Subsets: </i>MEDLINE
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        Value: 10.1016/j.slasd.2024.100162
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              Text: 2024 Jul
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