Design, synthesis and biological evaluation of arylsulfonamides as ADAMTS7 inhibitors.

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Title: Design, synthesis and biological evaluation of arylsulfonamides as ADAMTS7 inhibitors.
Authors: Cuffaro D; Department of Pharmacy, University of Pisa Via Bonanno 6 56126 Pisa Italy elisa.nuti@unipi.it +39 0502219551., Burkhard T; Department of Biochemical and Physiological Sciences, School of Biosciences, Faculty of Health and Medical Sciences, University of Surrey Edward Jenner Building Guildford GU2 7XH UK s.santamaria@surrey.ac.uk., Bernardoni BL; Department of Pharmacy, University of Pisa Via Bonanno 6 56126 Pisa Italy elisa.nuti@unipi.it +39 0502219551., Di Leo R; Department of Pharmacy, University of Pisa Via Bonanno 6 56126 Pisa Italy elisa.nuti@unipi.it +39 0502219551., Zhang X; Institute of Cardiovascular Science, University College London 51 Chenies Mews London WC1E 6HX UK R.deGroot@ucl.ac.uk +44 (0) 20 3108 1423., Galati S; Department of Pharmacy, University of Pisa Via Bonanno 6 56126 Pisa Italy elisa.nuti@unipi.it +39 0502219551., Tuccinardi T; Department of Pharmacy, University of Pisa Via Bonanno 6 56126 Pisa Italy elisa.nuti@unipi.it +39 0502219551., Macchia M; Department of Pharmacy, University of Pisa Via Bonanno 6 56126 Pisa Italy elisa.nuti@unipi.it +39 0502219551., Rossello A; Department of Pharmacy, University of Pisa Via Bonanno 6 56126 Pisa Italy elisa.nuti@unipi.it +39 0502219551., Santamaria S; Department of Biochemical and Physiological Sciences, School of Biosciences, Faculty of Health and Medical Sciences, University of Surrey Edward Jenner Building Guildford GU2 7XH UK s.santamaria@surrey.ac.uk., de Groot R; Institute of Cardiovascular Science, University College London 51 Chenies Mews London WC1E 6HX UK R.deGroot@ucl.ac.uk +44 (0) 20 3108 1423., Nuti E; Department of Pharmacy, University of Pisa Via Bonanno 6 56126 Pisa Italy elisa.nuti@unipi.it +39 0502219551.
Source: RSC medicinal chemistry [RSC Med Chem] 2024 Jun 19; Vol. 15 (8), pp. 2806-2825. Date of Electronic Publication: 2024 Jun 19 (Print Publication: 2024).
Publication Type: Journal Article
Journal Info: Publisher: Royal Society of Chemistry Country of Publication: England NLM ID: 101759460 Publication Model: eCollection Cited Medium: Internet ISSN: 2632-8682 (Electronic) Linking ISSN: 26328682 NLM ISO Abbreviation: RSC Med Chem Subsets: PubMed not MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:2632-8682
DOI:10.1039/d4md00149d