Identifying novel chemical matter against the Chikungunya virus nsP3 macrodomain through crystallographic fragment screening.

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Title: Identifying novel chemical matter against the Chikungunya virus nsP3 macrodomain through crystallographic fragment screening.
Authors: Aschenbrenner JC; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom., de Godoy AS; São Carlos Institute of Physics, University of São Paulo, São Carlos, Brazil., Fairhead M; Centre for Medicines Discovery, University of Oxford, Oxford, United Kingdom., Tomlinson CWE; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom., Winokan M; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom., Balcomb BH; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom., Capkin E; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom., Chandran AV; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom., Golding M; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom., Koekemoer L; Centre for Medicines Discovery, University of Oxford, Oxford, United Kingdom., Lithgo RM; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom., Marples PG; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom., Ni X; Centre for Medicines Discovery, University of Oxford, Oxford, United Kingdom., Thompson W; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom., Wild C; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom., Xavier ME; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom., Fearon D; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom., von Delft F; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Centre for Medicines Discovery, University of Oxford, Oxford, United Kingdom.; Department of Biochemistry, University of Johannesburg, Auckland Park, South Africa.
Source: BioRxiv : the preprint server for biology [bioRxiv] 2024 Aug 23. Date of Electronic Publication: 2024 Aug 23.
Publication Type: Journal Article; Preprint
Journal Info: Country of Publication: United States NLM ID: 101680187 Publication Model: Electronic Cited Medium: Internet ISSN: 2692-8205 (Electronic) Linking ISSN: 26928205 NLM ISO Abbreviation: bioRxiv Subsets: PubMed not MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:2692-8205
DOI:10.1101/2024.08.23.609196