Identifying novel chemical matter against the Chikungunya virus nsP3 macrodomain through crystallographic fragment screening.
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| Title: | Identifying novel chemical matter against the Chikungunya virus nsP3 macrodomain through crystallographic fragment screening. |
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| Authors: | Aschenbrenner JC; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom., de Godoy AS; São Carlos Institute of Physics, University of São Paulo, São Carlos, Brazil., Fairhead M; Centre for Medicines Discovery, University of Oxford, Oxford, United Kingdom., Tomlinson CWE; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom., Winokan M; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom., Balcomb BH; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom., Capkin E; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom., Chandran AV; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom., Golding M; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom., Koekemoer L; Centre for Medicines Discovery, University of Oxford, Oxford, United Kingdom., Lithgo RM; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom., Marples PG; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom., Ni X; Centre for Medicines Discovery, University of Oxford, Oxford, United Kingdom., Thompson W; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom., Wild C; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom., Xavier ME; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom., Fearon D; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom., von Delft F; Diamond Light Source, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Research Complex at Harwell, Harwell Science & Innovation Campus, Didcot, United Kingdom.; Centre for Medicines Discovery, University of Oxford, Oxford, United Kingdom.; Department of Biochemistry, University of Johannesburg, Auckland Park, South Africa. |
| Source: | BioRxiv : the preprint server for biology [bioRxiv] 2024 Aug 23. Date of Electronic Publication: 2024 Aug 23. |
| Publication Type: | Journal Article; Preprint |
| Journal Info: | Country of Publication: United States NLM ID: 101680187 Publication Model: Electronic Cited Medium: Internet ISSN: 2692-8205 (Electronic) Linking ISSN: 26928205 NLM ISO Abbreviation: bioRxiv Subsets: PubMed not MEDLINE |
| Database: | MEDLINE Ultimate |
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