Design, preparation and biological evaluation of new Rociletinib-inspired analogs as irreversible EGFR inhibitors to treat non-small-cell-lung cancer.

Saved in:
Bibliographic Details
Title: Design, preparation and biological evaluation of new Rociletinib-inspired analogs as irreversible EGFR inhibitors to treat non-small-cell-lung cancer.
Authors: Konsue A; Department of Biomedical Engineering, School of Engineering, King Mongkut's Institute of Technology Ladkrabang, Bangkok 10520, Thailand., Lamtha T; Department of Biochemistry, Faculty of Science, Kasetsart University, Bangkok 10900, Thailand., Gleeson D; Department of Chemistry & Applied Computational Chemistry Research Unit, School of Science, King Mongkut's Institute of Technology Ladkrabang, Bangkok 10520, Thailand., Jones DJL; Leicester Cancer Research Centre, University of Leicester, Leicester LE1 7RH, United Kingdom., Britton RG; Leicester Cancer Research Centre, University of Leicester, Leicester LE1 7RH, United Kingdom., Pickering JD; School of Chemistry, University of Leicester, Leicester LE1 7RH, United Kingdom., Choowongkomon K; Department of Biochemistry, Faculty of Science, Kasetsart University, Bangkok 10900, Thailand., Gleeson MP; Department of Biomedical Engineering, School of Engineering, King Mongkut's Institute of Technology Ladkrabang, Bangkok 10520, Thailand. Electronic address: paul.gl@kmitl.ac.th.
Source: Bioorganic & medicinal chemistry [Bioorg Med Chem] 2024 Nov 01; Vol. 113, pp. 117906. Date of Electronic Publication: 2024 Sep 07.
Publication Type: Journal Article
Journal Info: Publisher: Elsevier Science Country of Publication: England NLM ID: 9413298 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3391 (Electronic) Linking ISSN: 09680896 NLM ISO Abbreviation: Bioorg Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
FullText Text:
  Availability: 0
Header DbId: mdl
DbLabel: MEDLINE Ultimate
An: 39299082
AccessLevel: 2
PubType: Academic Journal
PubTypeId: academicJournal
PreciseRelevancyScore: 0
IllustrationInfo
Items – Name: Title
  Label: Title
  Group: Ti
  Data: Design, preparation and biological evaluation of new Rociletinib-inspired analogs as irreversible EGFR inhibitors to treat non-small-cell-lung cancer.
– Name: Author
  Label: Authors
  Group: Au
  Data: <searchLink fieldCode="AU" term="%22Konsue+A%22">Konsue A</searchLink>; Department of Biomedical Engineering, School of Engineering, King Mongkut's Institute of Technology Ladkrabang, Bangkok 10520, Thailand.<br /><searchLink fieldCode="AU" term="%22Lamtha+T%22">Lamtha T</searchLink>; Department of Biochemistry, Faculty of Science, Kasetsart University, Bangkok 10900, Thailand.<br /><searchLink fieldCode="AU" term="%22Gleeson+D%22">Gleeson D</searchLink>; Department of Chemistry & Applied Computational Chemistry Research Unit, School of Science, King Mongkut's Institute of Technology Ladkrabang, Bangkok 10520, Thailand.<br /><searchLink fieldCode="AU" term="%22Jones+DJL%22">Jones DJL</searchLink>; Leicester Cancer Research Centre, University of Leicester, Leicester LE1 7RH, United Kingdom.<br /><searchLink fieldCode="AU" term="%22Britton+RG%22">Britton RG</searchLink>; Leicester Cancer Research Centre, University of Leicester, Leicester LE1 7RH, United Kingdom.<br /><searchLink fieldCode="AU" term="%22Pickering+JD%22">Pickering JD</searchLink>; School of Chemistry, University of Leicester, Leicester LE1 7RH, United Kingdom.<br /><searchLink fieldCode="AU" term="%22Choowongkomon+K%22">Choowongkomon K</searchLink>; Department of Biochemistry, Faculty of Science, Kasetsart University, Bangkok 10900, Thailand.<br /><searchLink fieldCode="AU" term="%22Gleeson+MP%22">Gleeson MP</searchLink>; Department of Biomedical Engineering, School of Engineering, King Mongkut's Institute of Technology Ladkrabang, Bangkok 10520, Thailand. Electronic address: paul.gl@kmitl.ac.th.
– Name: TitleSource
  Label: Source
  Group: Src
  Data: <searchLink fieldCode="JN" term="%229413298%22">Bioorganic & medicinal chemistry</searchLink> [Bioorg Med Chem] 2024 Nov 01; Vol. 113, pp. 117906. <i>Date of Electronic Publication: </i>2024 Sep 07.
– Name: TypePub
  Label: Publication Type
  Group: TypPub
  Data: Journal Article
– Name: TitleSource
  Label: Journal Info
  Group: Src
  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Elsevier+Science%22">Elsevier Science </searchLink><i>Country of Publication: </i>England <i>NLM ID: </i>9413298 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1464-3391 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2209680896%22">09680896 </searchLink><i>NLM ISO Abbreviation: </i>Bioorg Med Chem <i>Subsets: </i>MEDLINE
PLink https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=39299082
RecordInfo BibRecord:
  BibEntity:
    Identifiers:
      – Type: doi
        Value: 10.1016/j.bmc.2024.117906
    Languages:
      – Code: eng
        Text: English
    PhysicalDescription:
      Pagination:
        StartPage: 117906
    Titles:
      – TitleFull: Design, preparation and biological evaluation of new Rociletinib-inspired analogs as irreversible EGFR inhibitors to treat non-small-cell-lung cancer.
        Type: main
  BibRelationships:
    HasContributorRelationships:
      – PersonEntity:
          Name:
            NameFull: Konsue A
      – PersonEntity:
          Name:
            NameFull: Lamtha T
      – PersonEntity:
          Name:
            NameFull: Gleeson D
      – PersonEntity:
          Name:
            NameFull: Jones DJL
      – PersonEntity:
          Name:
            NameFull: Britton RG
      – PersonEntity:
          Name:
            NameFull: Pickering JD
      – PersonEntity:
          Name:
            NameFull: Choowongkomon K
      – PersonEntity:
          Name:
            NameFull: Gleeson MP
    IsPartOfRelationships:
      – BibEntity:
          Dates:
            – D: 01
              M: 11
              Text: 2024 Nov 01
              Type: published
              Y: 2024
          Identifiers:
            – Type: issn-electronic
              Value: 1464-3391
          Numbering:
            – Type: volume
              Value: 113
          Titles:
            – TitleFull: Bioorganic & medicinal chemistry
              Type: main
ResultId 1