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Optimization of Potent and Selective Cyclohexyl Acid ERAP1 Inhibitors Using Structure- and Property-Based Drug Design.

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Title: Optimization of Potent and Selective Cyclohexyl Acid ERAP1 Inhibitors Using Structure- and Property-Based Drug Design.
Authors: Hryczanek RP; GSK, Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, U.K.; Department of Pure and Applied Chemistry, University of Strathclyde, Glasgow G1 1XL, U.K., Hackett AS; GSK, Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, U.K., Rowland P; GSK, Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, U.K., Chung CW; GSK, Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, U.K., Convery MA; GSK, Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, U.K., Holmes DS; GSK, Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, U.K., Hutchinson JP; GSK, Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, U.K., Kitchen S; GSK, Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, U.K., Korczynska J; GSK, Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, U.K., Law RP; GSK, Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, U.K., Lea JD; GSK, Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, U.K., Liddle J; GSK, Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, U.K., Lonsdale R; GSK, Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, U.K., Neu M; GSK, Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, U.K., Nickels L; GSK, Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, U.K., Phillipou A; GSK, Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, U.K., Rowedder JE; GSK, Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, U.K., Schneck JL; GSK, Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, U.K., Scott-Stevens P; GSK, Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, U.K., Sheehan H; GSK, Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, U.K., Tayler CL; GSK, Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, U.K., Temponeras I; National Center for Scientific Research 'Demokritos', Agia Paraskevi, Attiki 15341, Greece., Tinworth CP; GSK, Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, U.K., Walker AL; GSK, Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, U.K., Wojno-Picon J; GSK, Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, U.K., Young RJ; GSK, Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, U.K., Lindsay DM; Department of Pure and Applied Chemistry, University of Strathclyde, Glasgow G1 1XL, U.K., Stratikos E; National Center for Scientific Research 'Demokritos', Agia Paraskevi, Attiki 15341, Greece.
Source: ACS medicinal chemistry letters [ACS Med Chem Lett] 2024 Nov 06; Vol. 15 (12), pp. 2107-2114. Date of Electronic Publication: 2024 Nov 06 (Print Publication: 2024).
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1948-5875
DOI:10.1021/acsmedchemlett.4c00401