Optimizing Triglyceride Prodrugs of a Model Immunomodulator: Conjugation through the Phenol of Mycophenolic Acid (MPA) Markedly Promotes Lymphatic Drug Transport.
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| Title: | Optimizing Triglyceride Prodrugs of a Model Immunomodulator: Conjugation through the Phenol of Mycophenolic Acid (MPA) Markedly Promotes Lymphatic Drug Transport. |
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| Authors: | Hu L, Quach T; Seaport Therapeutics, 6 Tide Street, Boston, Massachusetts 02210, United States., Zheng D, Leong NJ, Sharma G, Lim SF, Bonner D; Seaport Therapeutics, 6 Tide Street, Boston, Massachusetts 02210, United States., Trevaskis NL, Simpson JS; Seaport Therapeutics, 6 Tide Street, Boston, Massachusetts 02210, United States., Han S, Porter CJH |
| Source: | Molecular pharmaceutics [Mol Pharm] 2025 Mar 03; Vol. 22 (3), pp. 1555-1567. Date of Electronic Publication: 2025 Feb 11. |
| Publication Type: | Journal Article; Research Support, Non-U.S. Gov't |
| Journal Info: | Publisher: American Chemical Society Country of Publication: United States NLM ID: 101197791 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1543-8392 (Electronic) Linking ISSN: 15438384 NLM ISO Abbreviation: Mol Pharm Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| ISSN: | 1543-8392 |
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| DOI: | 10.1021/acs.molpharmaceut.4c01272 |