PSKH1 kinase activity is differentially modulated via allosteric binding of Ca2+ sensor proteins.

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Bibliographic Details
Title: PSKH1 kinase activity is differentially modulated via allosteric binding of Ca2+ sensor proteins.
Authors: Horne CR; Walter and Eliza Hall Institute of Medical Research, Parkville, VIC 3052, Australia.; Department of Medical Biology, University of Melbourne, Parkville, VIC 3052, Australia.; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC 3052, Australia., Dite TA; Walter and Eliza Hall Institute of Medical Research, Parkville, VIC 3052, Australia.; Department of Medical Biology, University of Melbourne, Parkville, VIC 3052, Australia., Young SN; Walter and Eliza Hall Institute of Medical Research, Parkville, VIC 3052, Australia., Mather LJ; Walter and Eliza Hall Institute of Medical Research, Parkville, VIC 3052, Australia., Dagley LF; Walter and Eliza Hall Institute of Medical Research, Parkville, VIC 3052, Australia.; Department of Medical Biology, University of Melbourne, Parkville, VIC 3052, Australia., Johnson JL; Meyer Cancer Center, Weill Cornell Medicine, New York, NY 10021.; Department of Cell Biology, Harvard Medical School, Boston, MA 02115.; Dana-Farber Cancer Institute, Harvard Medical School, Boston, MA 02215., Yaron-Barir TM; Meyer Cancer Center, Weill Cornell Medicine, New York, NY 10021.; Englander Institute for Precision Medicine, Institute for Computational Biomedicine, Weill Cornell Medicine, New York, NY 10021.; Columbia University Vagelos College of Physicians and Surgeons, New York, NY 10032., Huntsman EM; Meyer Cancer Center, Weill Cornell Medicine, New York, NY 10021.; Englander Institute for Precision Medicine, Institute for Computational Biomedicine, Weill Cornell Medicine, New York, NY 10021., Daly LA; Department of Biochemistry, Cell and Systems Biology, Institute of Systems, Molecular and Integrative Biology, University of Liverpool, Liverpool L69 7ZB, United Kingdom.; Centre for Proteome Research, Institute of Systems, Molecular and Integrative Biology, University of Liverpool, Liverpool L69 7ZB, United Kingdom., Byrne DP; Department of Biochemistry, Cell and Systems Biology, Institute of Systems, Molecular and Integrative Biology, University of Liverpool, Liverpool L69 7ZB, United Kingdom., Cadell AL; Cancer Ecosystems Program, Garvan Institute of Medical Research, Sydney, NSW 2010, Australia., Ng BH; Cancer Ecosystems Program, Garvan Institute of Medical Research, Sydney, NSW 2010, Australia., Yousef J; Walter and Eliza Hall Institute of Medical Research, Parkville, VIC 3052, Australia.; Department of Medical Biology, University of Melbourne, Parkville, VIC 3052, Australia., Multari DH; Walter and Eliza Hall Institute of Medical Research, Parkville, VIC 3052, Australia.; Department of Medical Biology, University of Melbourne, Parkville, VIC 3052, Australia., Shen L; Walter and Eliza Hall Institute of Medical Research, Parkville, VIC 3052, Australia., McAloon LM; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC 3052, Australia.; School of Behavioural and Health Sciences, Australian Catholic University, Fitzroy, VIC 3065, Australia.; St. Vincent's Institute of Medical Research, Fitzroy, VIC 3065, Australia., Manning G; NuaBio Research, Burlingame, CA 94010., Febbraio MA; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC 3052, Australia., Means AR; Molecular and Cellular Biology, Baylor College of Medicine, Houston, TX 77030., Cantley LC; Meyer Cancer Center, Weill Cornell Medicine, New York, NY 10021.; Department of Cell Biology, Harvard Medical School, Boston, MA 02115.; Dana-Farber Cancer Institute, Harvard Medical School, Boston, MA 02215., Tanzer MC; Walter and Eliza Hall Institute of Medical Research, Parkville, VIC 3052, Australia.; Department of Medical Biology, University of Melbourne, Parkville, VIC 3052, Australia., Croucher DR; Cancer Ecosystems Program, Garvan Institute of Medical Research, Sydney, NSW 2010, Australia.; School of Clinical Medicine, Faculty of Medicine and Health, University of New South Wales Sydney, Sydney, NSW 2010, Australia., Eyers CE; Department of Biochemistry, Cell and Systems Biology, Institute of Systems, Molecular and Integrative Biology, University of Liverpool, Liverpool L69 7ZB, United Kingdom.; Centre for Proteome Research, Institute of Systems, Molecular and Integrative Biology, University of Liverpool, Liverpool L69 7ZB, United Kingdom., Eyers PA; Department of Biochemistry, Cell and Systems Biology, Institute of Systems, Molecular and Integrative Biology, University of Liverpool, Liverpool L69 7ZB, United Kingdom., Scott JW; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC 3052, Australia.; St. Vincent's Institute of Medical Research, Fitzroy, VIC 3065, Australia.; The Florey Institute of Neuroscience and Mental Health, Parkville, VIC 3052, Australia., Murphy JM; Walter and Eliza Hall Institute of Medical Research, Parkville, VIC 3052, Australia.; Department of Medical Biology, University of Melbourne, Parkville, VIC 3052, Australia.; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC 3052, Australia.
Source: Proceedings of the National Academy of Sciences of the United States of America [Proc Natl Acad Sci U S A] 2025 Feb 25; Vol. 122 (8), pp. e2420961122. Date of Electronic Publication: 2025 Feb 18.
Publication Type: Journal Article
Journal Info: Publisher: National Academy of Sciences Country of Publication: United States NLM ID: 7505876 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1091-6490 (Electronic) Linking ISSN: 00278424 NLM ISO Abbreviation: Proc Natl Acad Sci U S A Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1091-6490
DOI:10.1073/pnas.2420961122