Physiologically Based Pharmacokinetic Modeling of Phosphate Prodrugs─Case Studies: Fostemsavir and Fostamatinib.

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Title: Physiologically Based Pharmacokinetic Modeling of Phosphate Prodrugs─Case Studies: Fostemsavir and Fostamatinib.
Authors: Stamatopoulos K; Biopharmaceutics, DPD, MDS, GSK, Ware SG12 0DP, U.K., Mistry N; Biopharmaceutics, DPD, MDS, GSK, Ware SG12 0DP, U.K., Taskar K; Drug Metabolism and Pharmacokinetics, GSK, Stevenage SG1 2NY, U.K., Salem F; Drug Metabolism and Pharmacokinetics, GSK, Stevenage SG1 2NY, U.K., Butler JM; Biopharmaceutics, DPD, MDS, GSK, Ware SG12 0DP, U.K., Tompson D; Clinical Pharmacology Modelling and Simulation, GSK, Medicines Research Centre, Stevenage SG1 2NY, U.K.
Source: Molecular pharmaceutics [Mol Pharm] 2025 Apr 07; Vol. 22 (4), pp. 2168-2181. Date of Electronic Publication: 2025 Mar 26.
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101197791 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1543-8392 (Electronic) Linking ISSN: 15438384 NLM ISO Abbreviation: Mol Pharm Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1543-8392
DOI:10.1021/acs.molpharmaceut.4c01362