Coculture-Based Screening Revealed Selective Cytostatic Effects of Pyrazol-Azepinoindoles.

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Title: Coculture-Based Screening Revealed Selective Cytostatic Effects of Pyrazol-Azepinoindoles.
Authors: Skvortsov DA; Chemistry Department and AN Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, Leninskie Gory, Building 1/3 GSP-1, Moscow, 119991, Russian Federation., Zhirkina IV; Chemistry Department and AN Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, Leninskie Gory, Building 1/3 GSP-1, Moscow, 119991, Russian Federation., Ipatova DA; Chemistry Department and AN Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, Leninskie Gory, Building 1/3 GSP-1, Moscow, 119991, Russian Federation., Vasilyeva LA; Chemistry Department and AN Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, Leninskie Gory, Building 1/3 GSP-1, Moscow, 119991, Russian Federation., Ivanenkov YA; P. Hertsen Moscow Oncology Research Institute, Moscow, 3125284, Russian Federation.; The Federal State Unitary Enterprise Dukhov Automatics Research Institute, Moscow, 127055, Russian Federation., Rubtsova MP; Chemistry Department and AN Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, Leninskie Gory, Building 1/3 GSP-1, Moscow, 119991, Russian Federation., Kartsev VG; InterBioScreen Ltd., Chernogolovka, 142432, Russian Federation., Sergiev PV; Chemistry Department and AN Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, Leninskie Gory, Building 1/3 GSP-1, Moscow, 119991, Russian Federation.; Center of Molecular and Cellular Biology, Moscow, 121205, Russian Federation., Dontsova OA; Chemistry Department and AN Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, Leninskie Gory, Building 1/3 GSP-1, Moscow, 119991, Russian Federation.; Center of Molecular and Cellular Biology, Moscow, 121205, Russian Federation.
Source: ChemMedChem [ChemMedChem] 2025 Jun 17; Vol. 20 (12), pp. e202500052. Date of Electronic Publication: 2025 Apr 24.
Publication Type: Journal Article
Journal Info: Publisher: Wiley-VCH Country of Publication: Germany NLM ID: 101259013 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1860-7187 (Electronic) Linking ISSN: 18607179 NLM ISO Abbreviation: ChemMedChem Subsets: MEDLINE
Database: MEDLINE Ultimate
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ISSN:1860-7187
DOI:10.1002/cmdc.202500052