Coculture-Based Screening Revealed Selective Cytostatic Effects of Pyrazol-Azepinoindoles.

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Title: Coculture-Based Screening Revealed Selective Cytostatic Effects of Pyrazol-Azepinoindoles.
Authors: Skvortsov DA; Chemistry Department and AN Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, Leninskie Gory, Building 1/3 GSP-1, Moscow, 119991, Russian Federation., Zhirkina IV; Chemistry Department and AN Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, Leninskie Gory, Building 1/3 GSP-1, Moscow, 119991, Russian Federation., Ipatova DA; Chemistry Department and AN Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, Leninskie Gory, Building 1/3 GSP-1, Moscow, 119991, Russian Federation., Vasilyeva LA; Chemistry Department and AN Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, Leninskie Gory, Building 1/3 GSP-1, Moscow, 119991, Russian Federation., Ivanenkov YA; P. Hertsen Moscow Oncology Research Institute, Moscow, 3125284, Russian Federation.; The Federal State Unitary Enterprise Dukhov Automatics Research Institute, Moscow, 127055, Russian Federation., Rubtsova MP; Chemistry Department and AN Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, Leninskie Gory, Building 1/3 GSP-1, Moscow, 119991, Russian Federation., Kartsev VG; InterBioScreen Ltd., Chernogolovka, 142432, Russian Federation., Sergiev PV; Chemistry Department and AN Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, Leninskie Gory, Building 1/3 GSP-1, Moscow, 119991, Russian Federation.; Center of Molecular and Cellular Biology, Moscow, 121205, Russian Federation., Dontsova OA; Chemistry Department and AN Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, Leninskie Gory, Building 1/3 GSP-1, Moscow, 119991, Russian Federation.; Center of Molecular and Cellular Biology, Moscow, 121205, Russian Federation.
Source: ChemMedChem [ChemMedChem] 2025 Jun 17; Vol. 20 (12), pp. e202500052. Date of Electronic Publication: 2025 Apr 24.
Publication Type: Journal Article
Journal Info: Publisher: Wiley-VCH Country of Publication: Germany NLM ID: 101259013 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1860-7187 (Electronic) Linking ISSN: 18607179 NLM ISO Abbreviation: ChemMedChem Subsets: MEDLINE
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  Data: Coculture-Based Screening Revealed Selective Cytostatic Effects of Pyrazol-Azepinoindoles.
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  Data: <searchLink fieldCode="AU" term="%22Skvortsov+DA%22">Skvortsov DA</searchLink>; Chemistry Department and AN Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, Leninskie Gory, Building 1/3 GSP-1, Moscow, 119991, Russian Federation.<br /><searchLink fieldCode="AU" term="%22Zhirkina+IV%22">Zhirkina IV</searchLink>; Chemistry Department and AN Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, Leninskie Gory, Building 1/3 GSP-1, Moscow, 119991, Russian Federation.<br /><searchLink fieldCode="AU" term="%22Ipatova+DA%22">Ipatova DA</searchLink>; Chemistry Department and AN Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, Leninskie Gory, Building 1/3 GSP-1, Moscow, 119991, Russian Federation.<br /><searchLink fieldCode="AU" term="%22Vasilyeva+LA%22">Vasilyeva LA</searchLink>; Chemistry Department and AN Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, Leninskie Gory, Building 1/3 GSP-1, Moscow, 119991, Russian Federation.<br /><searchLink fieldCode="AU" term="%22Ivanenkov+YA%22">Ivanenkov YA</searchLink>; P. Hertsen Moscow Oncology Research Institute, Moscow, 3125284, Russian Federation.; The Federal State Unitary Enterprise Dukhov Automatics Research Institute, Moscow, 127055, Russian Federation.<br /><searchLink fieldCode="AU" term="%22Rubtsova+MP%22">Rubtsova MP</searchLink>; Chemistry Department and AN Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, Leninskie Gory, Building 1/3 GSP-1, Moscow, 119991, Russian Federation.<br /><searchLink fieldCode="AU" term="%22Kartsev+VG%22">Kartsev VG</searchLink>; InterBioScreen Ltd., Chernogolovka, 142432, Russian Federation.<br /><searchLink fieldCode="AU" term="%22Sergiev+PV%22">Sergiev PV</searchLink>; Chemistry Department and AN Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, Leninskie Gory, Building 1/3 GSP-1, Moscow, 119991, Russian Federation.; Center of Molecular and Cellular Biology, Moscow, 121205, Russian Federation.<br /><searchLink fieldCode="AU" term="%22Dontsova+OA%22">Dontsova OA</searchLink>; Chemistry Department and AN Belozersky Institute of Physico-Chemical Biology, Lomonosov Moscow State University, Leninskie Gory, Building 1/3 GSP-1, Moscow, 119991, Russian Federation.; Center of Molecular and Cellular Biology, Moscow, 121205, Russian Federation.
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  Data: <searchLink fieldCode="JN" term="%22101259013%22">ChemMedChem</searchLink> [ChemMedChem] 2025 Jun 17; Vol. 20 (12), pp. e202500052. <i>Date of Electronic Publication: </i>2025 Apr 24.
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              Text: 2025 Jun 17
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