A scaffold repositioning approach: dihydroBenzoImidazoTriazineDione (BITD) derivatives as selective ALDH1A1 inhibitors.
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| Title: | A scaffold repositioning approach: dihydroBenzoImidazoTriazineDione (BITD) derivatives as selective ALDH1A1 inhibitors. |
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| Authors: | Bernardoni BL; Department of Pharmacy, University of Pisa, 56126, Pisa, Italy., D'Agostino I; Department of Pharmacy, University of Pisa, 56126, Pisa, Italy. ilaria.dagostino@unipi.it., Siragusa S; Department of Pharmaceutical Sciences, University of Piemonte Orientale, 28100, Novara, Italy., Mori M; Department of Biotechnology, Chemistry and Pharmacy, University of Siena, 53100, Siena, Italy., Garavaglia S; Department of Pharmaceutical Sciences, University of Piemonte Orientale, 28100, Novara, Italy. silvia.garavaglia@uniupo.it., La Motta C; Department of Pharmacy, University of Pisa, 56126, Pisa, Italy. |
| Source: | Molecular diversity [Mol Divers] 2026 Feb; Vol. 30 (1), pp. 495-508. Date of Electronic Publication: 2025 Apr 04. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: ESCOM Science Publishers Country of Publication: Netherlands NLM ID: 9516534 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1573-501X (Electronic) Linking ISSN: 13811991 NLM ISO Abbreviation: Mol Divers Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
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| ISSN: | 1573-501X |
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| DOI: | 10.1007/s11030-025-11179-6 |