Applications of contemporary tools to measure plasma protein binding of targeted protein degraders.

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Bibliographic Details
Title: Applications of contemporary tools to measure plasma protein binding of targeted protein degraders.
Authors: Niosi M; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, Groton, Connecticut. Electronic address: Mark.Niosi@pfizer.com., Zhang S; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, Groton, Connecticut., Burchett W; Global Biometrics and Data Management, Pfizer Worldwide Research and Development, Groton, Connecticut., Heck CJS; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, Groton, Connecticut., Goetz GH; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, Groton, Connecticut., Federico JJ; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, Groton, Connecticut., Gernhardt S; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, Groton, Connecticut., Jordan S; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, Groton, Connecticut., Gilbert AM; Medicinal Chemistry, Pfizer Worldwide Research and Development, Groton, Connecticut., Calabrese MF; Discovery Sciences, Pfizer Worldwide Research and Development, Groton, Connecticut., Obach RS; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, Groton, Connecticut., Steyn SJ; Pharmacokinetics, Dynamics and Metabolism, Pfizer Worldwide Research and Development, Cambridge, Massachusetts.
Source: Drug metabolism and disposition: the biological fate of chemicals [Drug Metab Dispos] 2025 May; Vol. 53 (5), pp. 100066. Date of Electronic Publication: 2025 Mar 19.
Publication Type: Journal Article
Journal Info: Publisher: American Society for Pharmacology and Experimental Therapeutics, etc.] Country of Publication: Netherlands NLM ID: 9421550 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1521-009X (Electronic) Linking ISSN: 00909556 NLM ISO Abbreviation: Drug Metab Dispos Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1521-009X
DOI:10.1016/j.dmd.2025.100066