Compounds with dual glutaminase inhibition and Nrf2 activation activities enhance morphine analgesia and reduce pain sensitization in chemotherapy-induced peripheral neuropathy mouse model.

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Title: Compounds with dual glutaminase inhibition and Nrf2 activation activities enhance morphine analgesia and reduce pain sensitization in chemotherapy-induced peripheral neuropathy mouse model.
Authors: Foster BK; Department of Pharmaceutical and Graduate Life Sciences, College of Health Professions, Nursing & Pharmacy, Manchester University Fort Wayne, Fort Wayne, Indiana., Kliebe V; Darby Children's Research Institute, Department of Pediatrics, Medical University of South Carolina, Charleston, South Carolina., Elnaham HF; Department of Pharmaceutical and Graduate Life Sciences, College of Health Professions, Nursing & Pharmacy, Manchester University Fort Wayne, Fort Wayne, Indiana., Thompson MK; Department of Pharmaceutical and Graduate Life Sciences, College of Health Professions, Nursing & Pharmacy, Manchester University Fort Wayne, Fort Wayne, Indiana., Sagna SL; Department of Pharmaceutical and Graduate Life Sciences, College of Health Professions, Nursing & Pharmacy, Manchester University Fort Wayne, Fort Wayne, Indiana., Patton JS; Department of Pharmaceutical and Graduate Life Sciences, College of Health Professions, Nursing & Pharmacy, Manchester University Fort Wayne, Fort Wayne, Indiana., Brown SC; Department of Pharmaceutical and Graduate Life Sciences, College of Health Professions, Nursing & Pharmacy, Manchester University Fort Wayne, Fort Wayne, Indiana., Chen X; Department of Pharmaceutical and Clinical Sciences, College of Pharmacy and Health Sciences, Campbell University, Buies Creek, North Carolina., Liu T; Department of Biomedical Sciences, West Virginia School of Osteopathic Medicine, Lewisburg, West Virginia., Bowden J; Department of Pharmacology, College of Medicine, University of Arizona, Tuscon, Arizona., Streicher J; Department of Pharmacology, College of Medicine, University of Arizona, Tuscon, Arizona., Lei W; Department of Pharmaceutical and Graduate Life Sciences, College of Health Professions, Nursing & Pharmacy, Manchester University Fort Wayne, Fort Wayne, Indiana. Electronic address: wlei@manchester.edu.
Source: The Journal of pharmacology and experimental therapeutics [J Pharmacol Exp Ther] 2025 Jun; Vol. 392 (6), pp. 103583. Date of Electronic Publication: 2025 Apr 16.
Publication Type: Journal Article
Journal Info: Publisher: Elsevier Country of Publication: Netherlands NLM ID: 0376362 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1521-0103 (Electronic) Linking ISSN: 00223565 NLM ISO Abbreviation: J Pharmacol Exp Ther Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: Compounds with dual glutaminase inhibition and Nrf2 activation activities enhance morphine analgesia and reduce pain sensitization in chemotherapy-induced peripheral neuropathy mouse model.
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  Data: <searchLink fieldCode="AU" term="%22Foster+BK%22">Foster BK</searchLink>; Department of Pharmaceutical and Graduate Life Sciences, College of Health Professions, Nursing & Pharmacy, Manchester University Fort Wayne, Fort Wayne, Indiana.<br /><searchLink fieldCode="AU" term="%22Kliebe+V%22">Kliebe V</searchLink>; Darby Children's Research Institute, Department of Pediatrics, Medical University of South Carolina, Charleston, South Carolina.<br /><searchLink fieldCode="AU" term="%22Elnaham+HF%22">Elnaham HF</searchLink>; Department of Pharmaceutical and Graduate Life Sciences, College of Health Professions, Nursing & Pharmacy, Manchester University Fort Wayne, Fort Wayne, Indiana.<br /><searchLink fieldCode="AU" term="%22Thompson+MK%22">Thompson MK</searchLink>; Department of Pharmaceutical and Graduate Life Sciences, College of Health Professions, Nursing & Pharmacy, Manchester University Fort Wayne, Fort Wayne, Indiana.<br /><searchLink fieldCode="AU" term="%22Sagna+SL%22">Sagna SL</searchLink>; Department of Pharmaceutical and Graduate Life Sciences, College of Health Professions, Nursing & Pharmacy, Manchester University Fort Wayne, Fort Wayne, Indiana.<br /><searchLink fieldCode="AU" term="%22Patton+JS%22">Patton JS</searchLink>; Department of Pharmaceutical and Graduate Life Sciences, College of Health Professions, Nursing & Pharmacy, Manchester University Fort Wayne, Fort Wayne, Indiana.<br /><searchLink fieldCode="AU" term="%22Brown+SC%22">Brown SC</searchLink>; Department of Pharmaceutical and Graduate Life Sciences, College of Health Professions, Nursing & Pharmacy, Manchester University Fort Wayne, Fort Wayne, Indiana.<br /><searchLink fieldCode="AU" term="%22Chen+X%22">Chen X</searchLink>; Department of Pharmaceutical and Clinical Sciences, College of Pharmacy and Health Sciences, Campbell University, Buies Creek, North Carolina.<br /><searchLink fieldCode="AU" term="%22Liu+T%22">Liu T</searchLink>; Department of Biomedical Sciences, West Virginia School of Osteopathic Medicine, Lewisburg, West Virginia.<br /><searchLink fieldCode="AU" term="%22Bowden+J%22">Bowden J</searchLink>; Department of Pharmacology, College of Medicine, University of Arizona, Tuscon, Arizona.<br /><searchLink fieldCode="AU" term="%22Streicher+J%22">Streicher J</searchLink>; Department of Pharmacology, College of Medicine, University of Arizona, Tuscon, Arizona.<br /><searchLink fieldCode="AU" term="%22Lei+W%22">Lei W</searchLink>; Department of Pharmaceutical and Graduate Life Sciences, College of Health Professions, Nursing & Pharmacy, Manchester University Fort Wayne, Fort Wayne, Indiana. Electronic address: wlei@manchester.edu.
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  Data: <searchLink fieldCode="JN" term="%220376362%22">The Journal of pharmacology and experimental therapeutics</searchLink> [J Pharmacol Exp Ther] 2025 Jun; Vol. 392 (6), pp. 103583. <i>Date of Electronic Publication: </i>2025 Apr 16.
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Elsevier%22">Elsevier </searchLink><i>Country of Publication: </i>Netherlands <i>NLM ID: </i>0376362 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1521-0103 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2200223565%22">00223565 </searchLink><i>NLM ISO Abbreviation: </i>J Pharmacol Exp Ther <i>Subsets: </i>MEDLINE
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              Text: 2025 Jun
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