Recognition of the CREB-Binding Protein/Mixed Lineage Leukemia Interface by Sulfonyl-γ-AApeptides: Beyond Mimicry of Mixed Lineage Leukemia.

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Title: Recognition of the CREB-Binding Protein/Mixed Lineage Leukemia Interface by Sulfonyl-γ-AApeptides: Beyond Mimicry of Mixed Lineage Leukemia.
Authors: Huang B; Department of Chemistry, University of South Florida, Tampa, Florida 33620, United States., Wang M; Department of Chemistry, University of South Florida, Tampa, Florida 33620, United States., Gregory-Lott E; Department of Chemistry, University of South Florida, Tampa, Florida 33620, United States.; Department of Molecular Biosciences, University of South Florida, Tampa, Florida 33620, United States., Li BX; Program in Chemical Biology, Department of Chemical Physiology and Biochemistry, Oregon Health & Science University, Portland, Oregon 97239, United States.; Knight Cancer Institute, Oregon Health & Science University, Portland, Oregon 97239, United States., Win YY; Department of Chemistry, University of South Florida, Tampa, Florida 33620, United States., Shen N; Department of Chemistry, University of South Florida, Tampa, Florida 33620, United States.; Department of Pharmaceutical Sciences, University of South Florida, Tampa, Florida 33612, United States., Chen J; Department of Chemistry, University of South Florida, Tampa, Florida 33620, United States., Li S; Department of Chemistry, University of South Florida, Tampa, Florida 33620, United States., Cao C; Department of Pharmaceutical Sciences, University of South Florida, Tampa, Florida 33612, United States., Xiao X; Program in Chemical Biology, Department of Chemical Physiology and Biochemistry, Oregon Health & Science University, Portland, Oregon 97239, United States.; Knight Cancer Institute, Oregon Health & Science University, Portland, Oregon 97239, United States., Daughdrill GW; Department of Molecular Biosciences, University of South Florida, Tampa, Florida 33620, United States., Cai J; Department of Chemistry, University of South Florida, Tampa, Florida 33620, United States.
Source: Journal of medicinal chemistry [J Med Chem] 2025 Jun 12; Vol. 68 (11), pp. 12272-12283. Date of Electronic Publication: 2025 Jun 02.
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1520-4804
DOI:10.1021/acs.jmedchem.5c01148