Targeting protein disorder: the next hurdle in drug discovery.

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Title: Targeting protein disorder: the next hurdle in drug discovery.
Authors: Lazar T; VIB-VUB Center for Structural Biology, Vlaams Instituut voor Biotechnologie (VIB), Brussels, Belgium.; Structural Biology Brussels, Vrije Universiteit Brussel (VUB), Brussels, Belgium., Connor A; New Equilibrium Biosciences, Boston, MA, USA., DeLisle CF; New Equilibrium Biosciences, Boston, MA, USA., Burger V; New Equilibrium Biosciences, Boston, MA, USA. virginia@blackbirdlab.org.; Blackbird Laboratories, Baltimore, MD, USA. virginia@blackbirdlab.org., Tompa P; VIB-VUB Center for Structural Biology, Vlaams Instituut voor Biotechnologie (VIB), Brussels, Belgium. peter.tompa@vub.be.; Structural Biology Brussels, Vrije Universiteit Brussel (VUB), Brussels, Belgium. peter.tompa@vub.be.; New Equilibrium Biosciences, Boston, MA, USA. peter.tompa@vub.be.; Institute of Molecular Life Sciences, HUN-REN Research Centre for Natural Sciences (RCNS), Budapest, Hungary. peter.tompa@vub.be.; HUN-REN Office for Supported Research Groups (TKI), Cell Cycle Laboratory, National Institute of Oncology, Budapest, Hungary. peter.tompa@vub.be.
Source: Nature reviews. Drug discovery [Nat Rev Drug Discov] 2025 Oct; Vol. 24 (10), pp. 743-763. Date of Electronic Publication: 2025 Jun 09.
Publication Type: Journal Article; Review
Journal Info: Publisher: Nature Pub. Group Country of Publication: England NLM ID: 101124171 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1474-1784 (Electronic) Linking ISSN: 14741776 NLM ISO Abbreviation: Nat Rev Drug Discov Subsets: MEDLINE
Database: MEDLINE Ultimate
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ISSN:1474-1784
DOI:10.1038/s41573-025-01220-6