Design, evaluation, cytotoxic activity, molecular docking, ADMET analysis, and dynamic simulations and the preparation of new isoxazoles, thiazoles, 1,3-thiazines, and thiazolopyrimidines derived from quinoline-pyridopyrimidines.
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| Title: | Design, evaluation, cytotoxic activity, molecular docking, ADMET analysis, and dynamic simulations and the preparation of new isoxazoles, thiazoles, 1,3-thiazines, and thiazolopyrimidines derived from quinoline-pyridopyrimidines. |
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| Authors: | Abu-Hashem AA; Department of Physical Sciences, Chemistry Division, College of Science, Jazan University, Jazan, Saudi Arabia.; Photochemistry Department (Heterocyclic Unit), National Research Centre, Dokki, Egypt., Amri N; Department of Physical Sciences, Chemistry Division, College of Science, Jazan University, Jazan, Saudi Arabia., El-Sayed AF; Microbial Genetics Department, Biotechnology Research Institute, National Research Centre, Giza, Egypt.; Egypt Center for Research and Regenerative Medicine (ECRRM), Cairo, Egypt. |
| Source: | Pharmaceutical biology [Pharm Biol] 2025 Dec; Vol. 63 (1), pp. 607-644. Date of Electronic Publication: 2025 Aug 19. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: Taylor & Francis Country of Publication: England NLM ID: 9812552 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1744-5116 (Electronic) Linking ISSN: 13880209 NLM ISO Abbreviation: Pharm Biol Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
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| ISSN: | 1744-5116 |
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| DOI: | 10.1080/13880209.2025.2547744 |