Design, evaluation, cytotoxic activity, molecular docking, ADMET analysis, and dynamic simulations and the preparation of new isoxazoles, thiazoles, 1,3-thiazines, and thiazolopyrimidines derived from quinoline-pyridopyrimidines.

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Title: Design, evaluation, cytotoxic activity, molecular docking, ADMET analysis, and dynamic simulations and the preparation of new isoxazoles, thiazoles, 1,3-thiazines, and thiazolopyrimidines derived from quinoline-pyridopyrimidines.
Authors: Abu-Hashem AA; Department of Physical Sciences, Chemistry Division, College of Science, Jazan University, Jazan, Saudi Arabia.; Photochemistry Department (Heterocyclic Unit), National Research Centre, Dokki, Egypt., Amri N; Department of Physical Sciences, Chemistry Division, College of Science, Jazan University, Jazan, Saudi Arabia., El-Sayed AF; Microbial Genetics Department, Biotechnology Research Institute, National Research Centre, Giza, Egypt.; Egypt Center for Research and Regenerative Medicine (ECRRM), Cairo, Egypt.
Source: Pharmaceutical biology [Pharm Biol] 2025 Dec; Vol. 63 (1), pp. 607-644. Date of Electronic Publication: 2025 Aug 19.
Publication Type: Journal Article
Journal Info: Publisher: Taylor & Francis Country of Publication: England NLM ID: 9812552 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1744-5116 (Electronic) Linking ISSN: 13880209 NLM ISO Abbreviation: Pharm Biol Subsets: MEDLINE
Database: MEDLINE Ultimate
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ISSN:1744-5116
DOI:10.1080/13880209.2025.2547744