SAR Studies around the SULT1A1-Activated Alkylator YC-1 as Cytotoxic Agents against Biliary Tract Cancer Cells.

Saved in:
Bibliographic Details
Title: SAR Studies around the SULT1A1-Activated Alkylator YC-1 as Cytotoxic Agents against Biliary Tract Cancer Cells.
Authors: Kong K; National Center for Advancing Translational Science, National Institute of Health, 9800 Medical Center Drive, Rockville, Maryland 20850, United States., Zhao W; National Center for Advancing Translational Science, National Institute of Health, 9800 Medical Center Drive, Rockville, Maryland 20850, United States., Shrimp JH; National Center for Advancing Translational Science, National Institute of Health, 9800 Medical Center Drive, Rockville, Maryland 20850, United States., Vava M; National Center for Advancing Translational Science, National Institute of Health, 9800 Medical Center Drive, Rockville, Maryland 20850, United States., Sinha R; National Center for Advancing Translational Science, National Institute of Health, 9800 Medical Center Drive, Rockville, Maryland 20850, United States., Sharma S; National Center for Advancing Translational Science, National Institute of Health, 9800 Medical Center Drive, Rockville, Maryland 20850, United States., Lee TD; National Center for Advancing Translational Science, National Institute of Health, 9800 Medical Center Drive, Rockville, Maryland 20850, United States., Roth JS; National Center for Advancing Translational Science, National Institute of Health, 9800 Medical Center Drive, Rockville, Maryland 20850, United States., Lee OW; National Center for Advancing Translational Science, National Institute of Health, 9800 Medical Center Drive, Rockville, Maryland 20850, United States., Lewis D; National Center for Advancing Translational Science, National Institute of Health, 9800 Medical Center Drive, Rockville, Maryland 20850, United States., Kearney SE; National Center for Advancing Translational Science, National Institute of Health, 9800 Medical Center Drive, Rockville, Maryland 20850, United States., Rohde JM; National Center for Advancing Translational Science, National Institute of Health, 9800 Medical Center Drive, Rockville, Maryland 20850, United States., Davis MI; National Center for Advancing Translational Science, National Institute of Health, 9800 Medical Center Drive, Rockville, Maryland 20850, United States., Shah P; National Center for Advancing Translational Science, National Institute of Health, 9800 Medical Center Drive, Rockville, Maryland 20850, United States., Wang AQ; National Center for Advancing Translational Science, National Institute of Health, 9800 Medical Center Drive, Rockville, Maryland 20850, United States., Xu X; National Center for Advancing Translational Science, National Institute of Health, 9800 Medical Center Drive, Rockville, Maryland 20850, United States., Shi L; Massachusetts General Hospital Cancer Center, Harvard Medical School, Boston, Massachusetts 02114, United States., Shen M; National Center for Advancing Translational Science, National Institute of Health, 9800 Medical Center Drive, Rockville, Maryland 20850, United States., Boxer MB; National Center for Advancing Translational Science, National Institute of Health, 9800 Medical Center Drive, Rockville, Maryland 20850, United States., Bardeesy N; Massachusetts General Hospital Cancer Center, Harvard Medical School, Boston, Massachusetts 02114, United States., Hall MD; National Center for Advancing Translational Science, National Institute of Health, 9800 Medical Center Drive, Rockville, Maryland 20850, United States., Patnaik S; National Center for Advancing Translational Science, National Institute of Health, 9800 Medical Center Drive, Rockville, Maryland 20850, United States.
Source: Journal of medicinal chemistry [J Med Chem] 2025 Sep 25; Vol. 68 (18), pp. 18885-18907. Date of Electronic Publication: 2025 Sep 16.
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1520-4804
DOI:10.1021/acs.jmedchem.5c00489