2-Aminothiophene derivatives reduce resistance to fluoroquinolones in Staphylococcus aureus strains which overexpress NorA and MepA efflux pumps.

Saved in:
Bibliographic Details
Title: 2-Aminothiophene derivatives reduce resistance to fluoroquinolones in Staphylococcus aureus strains which overexpress NorA and MepA efflux pumps.
Authors: de Sousa Fernandes PA; Department of Biological Science, Laboratory of Synthesis and Drug Delivery-LSVM, State University of Paraiba, 58071-160, João Pessoa, PB, Brazil; Department of Pharmaceutical Sciences. Graduate Program in Natural and Synthetic Bioactive Products. Federal University of Paraiba, 58015-970, João Pessoa, PB, Brazil., de Araújo RSA; Department of Biological Science, Laboratory of Synthesis and Drug Delivery-LSVM, State University of Paraiba, 58071-160, João Pessoa, PB, Brazil; Department of Pharmaceutical Sciences. Graduate Program in Natural and Synthetic Bioactive Products. Federal University of Paraiba, 58015-970, João Pessoa, PB, Brazil., Gonçalves Alencar G; Department of Biological Chemistry. Laboratory of Microbiology and Molecular Biology-LMBM, Regional University of Cariri, 63105-000, Crato, CE, Brazil., Gonçalves SA; Department of Biological Chemistry. Laboratory of Microbiology and Molecular Biology-LMBM, Regional University of Cariri, 63105-000, Crato, CE, Brazil., de Araújo GA; Department of Biological Chemistry. Laboratory of Microbiology and Molecular Biology-LMBM, Regional University of Cariri, 63105-000, Crato, CE, Brazil., de Sousa Rodrigues EY; Department of Biological Chemistry. Laboratory of Microbiology and Molecular Biology-LMBM, Regional University of Cariri, 63105-000, Crato, CE, Brazil., Alves DS; Department of Biological Chemistry. Laboratory of Microbiology and Molecular Biology-LMBM, Regional University of Cariri, 63105-000, Crato, CE, Brazil., de Almeida RS; Department of Biological Chemistry. Laboratory of Microbiology and Molecular Biology-LMBM, Regional University of Cariri, 63105-000, Crato, CE, Brazil., de Morais Oliveira-Tintino CD; Department of Biological Chemistry. Laboratory of Microbiology and Molecular Biology-LMBM, Regional University of Cariri, 63105-000, Crato, CE, Brazil., Sidrônio MGS; Health Sciences Center. Graduate Program in Development and Technological Innovation in Medicines, Federal University of Paraiba, 58015-970, João Pessoa, PB, Brazil., Rodrigues VS; Department of Pharmaceutical Sciences. Graduate Program in Natural and Synthetic Bioactive Products. Federal University of Paraiba, 58015-970, João Pessoa, PB, Brazil., Araújo Padilha EK; Research Group on Biological and Molecular Chemistry, Institute of Chemistry and Biotechnology, Federal University of Alagoas, AC Simões campus, 57072-970, Maceió, Alagoas, Brazil., da Silva EF; Research Group on Biological and Molecular Chemistry, Institute of Chemistry and Biotechnology, Federal University of Alagoas, AC Simões campus, 57072-970, Maceió, Alagoas, Brazil., Nayarisseri A; In Silico Research Laboratory, Eminent Biosciences, Mahalakshmi Nagar, Indore, 452010, India., da Silva TG; Departament of Antibiotics, Federal University of Pernambuco, 50670-910, Recife, PE, Brazil., de Melo Coutinho HD; Department of Biological Chemistry. Laboratory of Microbiology and Molecular Biology-LMBM, Regional University of Cariri, 63105-000, Crato, CE, Brazil., Mendonça-Junior FJB; Department of Biological Science, Laboratory of Synthesis and Drug Delivery-LSVM, State University of Paraiba, 58071-160, João Pessoa, PB, Brazil; Department of Pharmaceutical Sciences. Graduate Program in Natural and Synthetic Bioactive Products. Federal University of Paraiba, 58015-970, João Pessoa, PB, Brazil. Electronic address: franciscojaime@servidor.uepb.edu.br.
Source: Biochimie [Biochimie] 2025 Dec; Vol. 239 (Pt B), pp. 191-206. Date of Electronic Publication: 2025 Sep 20.
Publication Type: Journal Article
Journal Info: Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 1264604 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1638-6183 (Electronic) Linking ISSN: 03009084 NLM ISO Abbreviation: Biochimie Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1638-6183
DOI:10.1016/j.biochi.2025.09.001