Revealing the rationale behind the differential neutralization of phospholipase A2 (PLA2) enzymes in snake and bee venom by varespladib (LY-315920), a small molecule PLA2 inhibitor.

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Title: Revealing the rationale behind the differential neutralization of phospholipase A2 (PLA2) enzymes in snake and bee venom by varespladib (LY-315920), a small molecule PLA2 inhibitor.
Authors: Kumar R; Division of Life Sciences, Institute of Advanced Study in Science and Technology, Vigyan Path, Garchuk, Guwahati, Assam, India.; Academy of Scientific and Innovative Research, AcSIR Headquarters CSIR-HRDC Campus, Postal Staff College Area, Ghaziabad, India., Patra A; Division of Life Sciences, Institute of Advanced Study in Science and Technology, Vigyan Path, Garchuk, Guwahati, Assam, India.; Amrita Research Centre, Amrita Vishwa Vidyapeetham, Faridabad, Haryana, India., Das D; Division of Life Sciences, Institute of Advanced Study in Science and Technology, Vigyan Path, Garchuk, Guwahati, Assam, India., Saikia K; Division of Life Sciences, Institute of Advanced Study in Science and Technology, Vigyan Path, Garchuk, Guwahati, Assam, India., da Silva JR; LAQV@REQUIMTE, Departamento de Química e Bioquímica, Faculdade De Ciências, Universidade do Porto, Porto, Portugal., Ramos MJ; LAQV@REQUIMTE, Departamento de Química e Bioquímica, Faculdade De Ciências, Universidade do Porto, Porto, Portugal., Khan MR; Division of Life Sciences, Institute of Advanced Study in Science and Technology, Vigyan Path, Garchuk, Guwahati, Assam, India.; Academy of Scientific and Innovative Research, AcSIR Headquarters CSIR-HRDC Campus, Postal Staff College Area, Ghaziabad, India., Fernandes PA; LAQV@REQUIMTE, Departamento de Química e Bioquímica, Faculdade De Ciências, Universidade do Porto, Porto, Portugal., Mukherjee AK; Division of Life Sciences, Institute of Advanced Study in Science and Technology, Vigyan Path, Garchuk, Guwahati, Assam, India.; Academy of Scientific and Innovative Research, AcSIR Headquarters CSIR-HRDC Campus, Postal Staff College Area, Ghaziabad, India.; Department of Molecular Biology and Biotechnology, Tezpur University, Tezpur, Assam, India.
Source: Journal of biomolecular structure & dynamics [J Biomol Struct Dyn] 2025 Dec 03, pp. 1-23. Date of Electronic Publication: 2025 Dec 03.
Publication Type: Journal Article
Journal Info: Publisher: Taylor & Francis Country of Publication: England NLM ID: 8404176 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1538-0254 (Electronic) Linking ISSN: 07391102 NLM ISO Abbreviation: J Biomol Struct Dyn Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1538-0254
DOI:10.1080/07391102.2025.2592598