Evaluation of Bifunctional, PSMA-Targeted Triazamacrocycle-Picolinates Compatible with the 18F/44Sc/177Lu Isotope Triad.

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Title: Evaluation of Bifunctional, PSMA-Targeted Triazamacrocycle-Picolinates Compatible with the 18F/44Sc/177Lu Isotope Triad.
Authors: Glaser OM; Department of Chemistry, University of Wisconsin-Madison, 1101 University Avenue, Madison, Wisconsin 53705, United States., Goerlach H; Department of Chemistry, University of Wisconsin-Madison, 1101 University Avenue, Madison, Wisconsin 53705, United States., Salek MV; Department of Medical Physics, University of Wisconsin-Madison, 1111 Highland Avenue, Madison, Wisconsin 53705, United States., Aluicio-Sarduy E; Department of Medical Physics, University of Wisconsin-Madison, 1111 Highland Avenue, Madison, Wisconsin 53705, United States., Gork MJ; Department of Chemistry, University of Wisconsin-Madison, 1101 University Avenue, Madison, Wisconsin 53705, United States., Śmiłowicz D; Department of Chemistry, University of Wisconsin-Madison, 1101 University Avenue, Madison, Wisconsin 53705, United States., Amason E; Department of Chemistry, University of Wisconsin-Madison, 1101 University Avenue, Madison, Wisconsin 53705, United States., Mixdorf JC; Department of Medical Physics, University of Wisconsin-Madison, 1111 Highland Avenue, Madison, Wisconsin 53705, United States., Barnhart TE; Department of Medical Physics, University of Wisconsin-Madison, 1111 Highland Avenue, Madison, Wisconsin 53705, United States., Engle JW; Department of Medical Physics, University of Wisconsin-Madison, 1111 Highland Avenue, Madison, Wisconsin 53705, United States.; Department of Radiology, University of Wisconsin-Madison, Madison, Wisconsin 53705, United States., Boros E; Department of Chemistry, University of Wisconsin-Madison, 1101 University Avenue, Madison, Wisconsin 53705, United States.
Source: Journal of medicinal chemistry [J Med Chem] 2025 Dec 25; Vol. 68 (24), pp. 26234-26245. Date of Electronic Publication: 2025 Dec 08.
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE
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  Data: Evaluation of Bifunctional, PSMA-Targeted Triazamacrocycle-Picolinates Compatible with the <superscript>18</superscript>F/<superscript>44</superscript>Sc/<superscript>177</superscript>Lu Isotope Triad.
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  Data: <searchLink fieldCode="AU" term="%22Glaser+OM%22">Glaser OM</searchLink>; Department of Chemistry, University of Wisconsin-Madison, 1101 University Avenue, Madison, Wisconsin 53705, United States.<br /><searchLink fieldCode="AU" term="%22Goerlach+H%22">Goerlach H</searchLink>; Department of Chemistry, University of Wisconsin-Madison, 1101 University Avenue, Madison, Wisconsin 53705, United States.<br /><searchLink fieldCode="AU" term="%22Salek+MV%22">Salek MV</searchLink>; Department of Medical Physics, University of Wisconsin-Madison, 1111 Highland Avenue, Madison, Wisconsin 53705, United States.<br /><searchLink fieldCode="AU" term="%22Aluicio-Sarduy+E%22">Aluicio-Sarduy E</searchLink>; Department of Medical Physics, University of Wisconsin-Madison, 1111 Highland Avenue, Madison, Wisconsin 53705, United States.<br /><searchLink fieldCode="AU" term="%22Gork+MJ%22">Gork MJ</searchLink>; Department of Chemistry, University of Wisconsin-Madison, 1101 University Avenue, Madison, Wisconsin 53705, United States.<br /><searchLink fieldCode="AU" term="%22Śmiłowicz+D%22">Śmiłowicz D</searchLink>; Department of Chemistry, University of Wisconsin-Madison, 1101 University Avenue, Madison, Wisconsin 53705, United States.<br /><searchLink fieldCode="AU" term="%22Amason+E%22">Amason E</searchLink>; Department of Chemistry, University of Wisconsin-Madison, 1101 University Avenue, Madison, Wisconsin 53705, United States.<br /><searchLink fieldCode="AU" term="%22Mixdorf+JC%22">Mixdorf JC</searchLink>; Department of Medical Physics, University of Wisconsin-Madison, 1111 Highland Avenue, Madison, Wisconsin 53705, United States.<br /><searchLink fieldCode="AU" term="%22Barnhart+TE%22">Barnhart TE</searchLink>; Department of Medical Physics, University of Wisconsin-Madison, 1111 Highland Avenue, Madison, Wisconsin 53705, United States.<br /><searchLink fieldCode="AU" term="%22Engle+JW%22">Engle JW</searchLink>; Department of Medical Physics, University of Wisconsin-Madison, 1111 Highland Avenue, Madison, Wisconsin 53705, United States.; Department of Radiology, University of Wisconsin-Madison, Madison, Wisconsin 53705, United States.<br /><searchLink fieldCode="AU" term="%22Boros+E%22">Boros E</searchLink>; Department of Chemistry, University of Wisconsin-Madison, 1101 University Avenue, Madison, Wisconsin 53705, United States.
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  Data: <searchLink fieldCode="JN" term="%229716531%22">Journal of medicinal chemistry</searchLink> [J Med Chem] 2025 Dec 25; Vol. 68 (24), pp. 26234-26245. <i>Date of Electronic Publication: </i>2025 Dec 08.
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