Genetic evidence for PARP1 trapping as a driver of PARP inhibitor efficacy in BRCA mutant cancer cells.

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Title: Genetic evidence for PARP1 trapping as a driver of PARP inhibitor efficacy in BRCA mutant cancer cells.
Authors: Ribeiro J; OTD Bioscience, Early Oncology, AstraZeneca, CambridgeCB20AA, United Kingdom., Hansen K; Discovery Sciences, R&D, AstraZeneca, CambridgeCB20AA,United Kingdom., van Beek L; Discovery Sciences, R&D, AstraZeneca, CambridgeCB20AA,United Kingdom., Stubbs C; Discovery Sciences, R&D, AstraZeneca, CambridgeCB20AA,United Kingdom., Frigola J; Oncology Data Science, Oncology R&D, AstraZeneca, CambridgeCB20AA,United Kingdom., Talbot S; OTD Bioscience, Early Oncology, AstraZeneca, CambridgeCB20AA, United Kingdom., Bentouati S; OTD Bioscience, Early Oncology, AstraZeneca, CambridgeCB20AA, United Kingdom., Hall J; OTD Bioscience, Early Oncology, AstraZeneca, CambridgeCB20AA, United Kingdom., Wijnhoven PWG; OTD Bioscience, Early Oncology, AstraZeneca, CambridgeCB20AA, United Kingdom., Armenia J; Oncology Data Science, Oncology R&D, AstraZeneca, CambridgeCB20AA,United Kingdom., Schimpl M; Discovery Sciences, R&D, AstraZeneca, CambridgeCB20AA,United Kingdom., Forment JV; OTD Bioscience, Early Oncology, AstraZeneca, CambridgeCB20AA, United Kingdom., Albertella MR; OTD Bioscience, Early Oncology, AstraZeneca, CambridgeCB20AA, United Kingdom., O'Connor MJ; OTD Bioscience, Early Oncology, AstraZeneca, CambridgeCB20AA, United Kingdom., Illuzzi G; OTD Bioscience, Early Oncology, AstraZeneca, CambridgeCB20AA, United Kingdom.
Source: Nucleic acids research [Nucleic Acids Res] 2025 Nov 26; Vol. 53 (22).
Publication Type: Journal Article
Journal Info: Publisher: Oxford University Press Country of Publication: England NLM ID: 0411011 Publication Model: Print Cited Medium: Internet ISSN: 1362-4962 (Electronic) Linking ISSN: 03051048 NLM ISO Abbreviation: Nucleic Acids Res Subsets: MEDLINE
Database: MEDLINE Ultimate
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Description
ISSN:1362-4962
DOI:10.1093/nar/gkaf1398