Discovery and Characterization of Zelnecirnon (RPT193), a Potent and Selective CCR4 Antagonist for Allergic Disorders.

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Bibliographic Details
Title: Discovery and Characterization of Zelnecirnon (RPT193), a Potent and Selective CCR4 Antagonist for Allergic Disorders.
Authors: Zibinsky M; RAPT Therapeutics, 561 Eccles Avenue, South San Francisco, California 94080, United States., Bradford D; RAPT Therapeutics, 561 Eccles Avenue, South San Francisco, California 94080, United States., Brockstedt DG; RAPT Therapeutics, 561 Eccles Avenue, South San Francisco, California 94080, United States., Corriden R; RAPT Therapeutics, 561 Eccles Avenue, South San Francisco, California 94080, United States., Jackson J; RAPT Therapeutics, 561 Eccles Avenue, South San Francisco, California 94080, United States., Jacobson S; RAPT Therapeutics, 561 Eccles Avenue, South San Francisco, California 94080, United States., Jiao S; RAPT Therapeutics, 561 Eccles Avenue, South San Francisco, California 94080, United States., Kassner PD; RAPT Therapeutics, 561 Eccles Avenue, South San Francisco, California 94080, United States., Ketcham JM; RAPT Therapeutics, 561 Eccles Avenue, South San Francisco, California 94080, United States., Marshall L; RAPT Therapeutics, 561 Eccles Avenue, South San Francisco, California 94080, United States., Okano A; RAPT Therapeutics, 561 Eccles Avenue, South San Francisco, California 94080, United States., Robles O; RAPT Therapeutics, 561 Eccles Avenue, South San Francisco, California 94080, United States., Schwarz J; RAPT Therapeutics, 561 Eccles Avenue, South San Francisco, California 94080, United States., Talay O; RAPT Therapeutics, 561 Eccles Avenue, South San Francisco, California 94080, United States., Tivitmahaisoon P; RAPT Therapeutics, 561 Eccles Avenue, South San Francisco, California 94080, United States., Lester-Zeiner D; RAPT Therapeutics, 561 Eccles Avenue, South San Francisco, California 94080, United States., Milestone H; RAPT Therapeutics, 561 Eccles Avenue, South San Francisco, California 94080, United States., Trujillo D; RAPT Therapeutics, 561 Eccles Avenue, South San Francisco, California 94080, United States., Younai A; RAPT Therapeutics, 561 Eccles Avenue, South San Francisco, California 94080, United States., Wustrow DJ; RAPT Therapeutics, 561 Eccles Avenue, South San Francisco, California 94080, United States.
Source: Journal of medicinal chemistry [J Med Chem] 2026 Feb 12; Vol. 69 (3), pp. 1982-1998. Date of Electronic Publication: 2026 Jan 23.
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1520-4804
DOI:10.1021/acs.jmedchem.5c01678