The Sigma1 receptor antagonist CM304 potentiates the antinociceptive effects of the cannabinoid receptor agonist delta9-tetrahydrocannabinol in rats and mice.

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Title: The Sigma1 receptor antagonist CM304 potentiates the antinociceptive effects of the cannabinoid receptor agonist delta9-tetrahydrocannabinol in rats and mice.
Authors: Zolali E; Department of Pharmaceutical Sciences, Jerry H. Hodge School of Pharmacy, Texas Tech University Health Sciences Center, Amarillo, TX, 79106, USA., Burns M; Department of Medicinal Chemistry, College of Pharmacy, University of Florida, 1225 Center Drive, PO Box 100484, Gainesville, FL, 32610, USA., Intagliata S; Department of Medicinal Chemistry, College of Pharmacy, University of Florida, 1225 Center Drive, PO Box 100484, Gainesville, FL, 32610, USA.; Department of Drug and Health Sciences, University of Catania, viale A. Doria 6, Catania, 95125, Italy., Patel A; Department of Pharmacodynamics, College of Pharmacy, University of Florida, Gainesville, FL, 32610, USA., Ho NP; Department of Pharmacodynamics, College of Pharmacy, University of Florida, Gainesville, FL, 32610, USA., Restrepo LF; Department of Pharmacodynamics, College of Pharmacy, University of Florida, Gainesville, FL, 32610, USA., Gamez-Jimenez LR; Department of Pharmacodynamics, College of Pharmacy, University of Florida, Gainesville, FL, 32610, USA., Alvarez MA; Department of Pharmacodynamics, College of Pharmacy, University of Florida, Gainesville, FL, 32610, USA., Wilson LL; Department of Pharmacodynamics, College of Pharmacy, University of Florida, Gainesville, FL, 32610, USA., Cutler SJ; College of Pharmacy, University of South Carolina, Columbia, SC, 29208, USA., McMahon LR; Department of Pharmaceutical Sciences, Jerry H. Hodge School of Pharmacy, Texas Tech University Health Sciences Center, Amarillo, TX, 79106, USA.; Department of Pharmacodynamics, College of Pharmacy, University of Florida, Gainesville, FL, 32610, USA., Hiranita T; Department of Drug and Health Sciences, University of Catania, viale A. Doria 6, Catania, 95125, Italy.; Department of Pharmacology, Joe R. and Teresa Lozano Long School of Medicine, University of Texas Health San Antonio, San Antonio, TX, 78229, USA., Obeng S; Department of Pharmaceutical Sciences, Jerry H. Hodge School of Pharmacy, Texas Tech University Health Sciences Center, Amarillo, TX, 79106, USA.; Department of Pharmacodynamics, College of Pharmacy, University of Florida, Gainesville, FL, 32610, USA., McCurdy CR; Department of Medicinal Chemistry, College of Pharmacy, University of Florida, 1225 Center Drive, PO Box 100484, Gainesville, FL, 32610, USA. CMccurdy@cop.ufl.edu.; Translational Drug Development Core, Clinical and Translational Sciences Institute, University of Florida, Gainesville, FL, 32610, USA. CMccurdy@cop.ufl.edu.
Source: Pharmacological reports : PR [Pharmacol Rep] 2026 Apr; Vol. 78 (2), pp. 431-445. Date of Electronic Publication: 2026 Feb 09.
Publication Type: Journal Article
Journal Info: Publisher: Springer International Publishing Country of Publication: Switzerland NLM ID: 101234999 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2299-5684 (Electronic) Linking ISSN: 17341140 NLM ISO Abbreviation: Pharmacol Rep Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:2299-5684
DOI:10.1007/s43440-026-00834-w