Mislocalisation of FLT3-ITD receptor contributes to MV4-11 leukaemia cell resistance to antibody-drug conjugate.

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Title: Mislocalisation of FLT3-ITD receptor contributes to MV4-11 leukaemia cell resistance to antibody-drug conjugate.
Authors: Nirachonkul W; Department of Medical Technology, Chiang Mai University, Chiang Mai, Thailand., Farrell MP; Department of Medicinal Chemistry, The University of Kansas, Lawrence, KS, USA., Tolbert TJ; Department of Pharmaceutical Chemistry, The University of Kansas, Lawrence, KS, USA., Okonogi S; Department of Pharmaceutical Sciences, Chiang Mai University, Chiang Mai, Thailand.; Center of Excellence in Pharmaceutical Nanotechnology, Chiang Mai University, Chiang Mai, Thailand., Tima S; Department of Medical Technology, Chiang Mai University, Chiang Mai, Thailand.; Center of Excellence in Pharmaceutical Nanotechnology, Chiang Mai University, Chiang Mai, Thailand.; Cancer Research Unit of Associated Medical Sciences (AMS CRU), Chiang Mai University, Thailand., Anuchapreeda S; Department of Medical Technology, Chiang Mai University, Chiang Mai, Thailand.; Center of Excellence in Pharmaceutical Nanotechnology, Chiang Mai University, Chiang Mai, Thailand.; Cancer Research Unit of Associated Medical Sciences (AMS CRU), Chiang Mai University, Thailand., Chiampanichayakul S; Department of Medical Technology, Chiang Mai University, Chiang Mai, Thailand.; Center of Excellence in Pharmaceutical Nanotechnology, Chiang Mai University, Chiang Mai, Thailand.; Cancer Research Unit of Associated Medical Sciences (AMS CRU), Chiang Mai University, Thailand., Siahaan TJ; Department of Pharmaceutical Chemistry, The University of Kansas, Lawrence, KS, USA.
Source: Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2026 Dec; Vol. 41 (1), pp. 2638027. Date of Electronic Publication: 2026 Mar 05.
Publication Type: Journal Article
Journal Info: Publisher: Taylor & Francis Country of Publication: England NLM ID: 101150203 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1475-6374 (Electronic) Linking ISSN: 14756366 NLM ISO Abbreviation: J Enzyme Inhib Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1475-6374
DOI:10.1080/14756366.2026.2638027