Discovery of Triazine-Based Toll-Like Receptor 9 Antagonists with Oral Activity.

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Bibliographic Details
Title: Discovery of Triazine-Based Toll-Like Receptor 9 Antagonists with Oral Activity.
Authors: Mandler MD; Bristol Myers Squibb Research, Princeton, New Jersey 08543, United States., Zhu Y; Bristol Myers Squibb Research, Princeton, New Jersey 08543, United States., Hollenbeck EC; Bristol Myers Squibb Research, Brisbane, California 94005, United States., Ziegler M; Bristol Myers Squibb Research, Princeton, New Jersey 08543, United States., Posy SL; Bristol Myers Squibb Research, Princeton, New Jersey 08543, United States., Mukundan S; Bristol Myers Squibb Research, Princeton, New Jersey 08543, United States., Halpern OS; Bristol Myers Squibb Research, Princeton, New Jersey 08543, United States., Driscoll JP; Bristol Myers Squibb Research, Brisbane, California 94005, United States., Wang T; Bristol Myers Squibb Research, Princeton, New Jersey 08543, United States., Huang L; Bristol Myers Squibb Research, Princeton, New Jersey 08543, United States., Fernando G; Bristol Myers Squibb Research, Princeton, New Jersey 08543, United States., Jung H; Bristol Myers Squibb Research, Princeton, New Jersey 08543, United States., Li L; Bristol Myers Squibb Research, Princeton, New Jersey 08543, United States., Cutrone J; Bristol Myers Squibb Research, Princeton, New Jersey 08543, United States., Baswar D; Biocon Bristol Myers Squibb R&D Centre, Bangalore 560100, India., Eapen P; Biocon Bristol Myers Squibb R&D Centre, Bangalore 560100, India., Traeger SC; Bristol Myers Squibb Research, Princeton, New Jersey 08543, United States., Srivastava S; Bristol Myers Squibb Research, Princeton, New Jersey 08543, United States., Olsen J; Bristol Myers Squibb Research, Princeton, New Jersey 08543, United States., Everlof GG; Bristol Myers Squibb Research, Princeton, New Jersey 08543, United States., Trujillo G; Bristol Myers Squibb Research, Princeton, New Jersey 08543, United States., Ellsworth BA; Bristol Myers Squibb Research, Princeton, New Jersey 08543, United States., Regueiro-Ren A; Bristol Myers Squibb Research, Princeton, New Jersey 08543, United States.
Source: ACS medicinal chemistry letters [ACS Med Chem Lett] 2026 Feb 27; Vol. 17 (3), pp. 727-732. Date of Electronic Publication: 2026 Feb 27 (Print Publication: 2026).
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1948-5875
DOI:10.1021/acsmedchemlett.5c00760