Synthesis, Radiochemistry, and Preclinical Assessment of the First GPR39 PET Imaging Agent.

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Bibliographic Details
Title: Synthesis, Radiochemistry, and Preclinical Assessment of the First GPR39 PET Imaging Agent.
Authors: Bhoopal B; Department of Radiology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States., Gollapelli KK; Department of Radiology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States., Damuka N; Department of Radiology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States., Krizan I; Department of Radiology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States., Miller M; Department of Radiology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States., Fitzgerald RW; Department of Radiology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States., Amesar N; Department of Radiology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States., Mumbaraddi D; Department of Chemistry, Wake Forest University, Winston-Salem, North Carolina 27109, United States., Zhu D; Department of Translational Neuroscience, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States., Cervera-Juanes R; Department of Translational Neuroscience, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States., Jadiya P; Department of Gerontology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States., Whitlow CT; Department of Radiology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States., Solingapuram Sai KK; Department of Radiology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States.
Source: Journal of medicinal chemistry [J Med Chem] 2026 Apr 09; Vol. 69 (7), pp. 7933-7944. Date of Electronic Publication: 2026 Mar 18.
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1520-4804
DOI:10.1021/acs.jmedchem.5c03351