Synthesis, Radiochemistry, and Preclinical Assessment of the First GPR39 PET Imaging Agent.

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Title: Synthesis, Radiochemistry, and Preclinical Assessment of the First GPR39 PET Imaging Agent.
Authors: Bhoopal B; Department of Radiology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States., Gollapelli KK; Department of Radiology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States., Damuka N; Department of Radiology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States., Krizan I; Department of Radiology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States., Miller M; Department of Radiology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States., Fitzgerald RW; Department of Radiology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States., Amesar N; Department of Radiology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States., Mumbaraddi D; Department of Chemistry, Wake Forest University, Winston-Salem, North Carolina 27109, United States., Zhu D; Department of Translational Neuroscience, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States., Cervera-Juanes R; Department of Translational Neuroscience, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States., Jadiya P; Department of Gerontology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States., Whitlow CT; Department of Radiology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States., Solingapuram Sai KK; Department of Radiology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States.
Source: Journal of medicinal chemistry [J Med Chem] 2026 Apr 09; Vol. 69 (7), pp. 7933-7944. Date of Electronic Publication: 2026 Mar 18.
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE
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  Data: <searchLink fieldCode="AU" term="%22Bhoopal+B%22">Bhoopal B</searchLink>; Department of Radiology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States.<br /><searchLink fieldCode="AU" term="%22Gollapelli+KK%22">Gollapelli KK</searchLink>; Department of Radiology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States.<br /><searchLink fieldCode="AU" term="%22Damuka+N%22">Damuka N</searchLink>; Department of Radiology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States.<br /><searchLink fieldCode="AU" term="%22Krizan+I%22">Krizan I</searchLink>; Department of Radiology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States.<br /><searchLink fieldCode="AU" term="%22Miller+M%22">Miller M</searchLink>; Department of Radiology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States.<br /><searchLink fieldCode="AU" term="%22Fitzgerald+RW%22">Fitzgerald RW</searchLink>; Department of Radiology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States.<br /><searchLink fieldCode="AU" term="%22Amesar+N%22">Amesar N</searchLink>; Department of Radiology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States.<br /><searchLink fieldCode="AU" term="%22Mumbaraddi+D%22">Mumbaraddi D</searchLink>; Department of Chemistry, Wake Forest University, Winston-Salem, North Carolina 27109, United States.<br /><searchLink fieldCode="AU" term="%22Zhu+D%22">Zhu D</searchLink>; Department of Translational Neuroscience, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States.<br /><searchLink fieldCode="AU" term="%22Cervera-Juanes+R%22">Cervera-Juanes R</searchLink>; Department of Translational Neuroscience, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States.<br /><searchLink fieldCode="AU" term="%22Jadiya+P%22">Jadiya P</searchLink>; Department of Gerontology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States.<br /><searchLink fieldCode="AU" term="%22Whitlow+CT%22">Whitlow CT</searchLink>; Department of Radiology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States.<br /><searchLink fieldCode="AU" term="%22Solingapuram+Sai+KK%22">Solingapuram Sai KK</searchLink>; Department of Radiology, Wake Forest School of Medicine, Winston-Salem, North Carolina 27157, United States.
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  Data: <searchLink fieldCode="JN" term="%229716531%22">Journal of medicinal chemistry</searchLink> [J Med Chem] 2026 Apr 09; Vol. 69 (7), pp. 7933-7944. <i>Date of Electronic Publication: </i>2026 Mar 18.
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