Development of SYK NanoBRET cellular target engagement assays for gain-of-function variants.

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Bibliographic Details
Title: Development of SYK NanoBRET cellular target engagement assays for gain-of-function variants.
Authors: Capener JL; Structural Genomics Consortium, Division of Chemical Biology and Medicinal Chemistry, Eshelman School of Pharmacy, The University of North Carolina at Chapel Hill, Chapel Hill, NC, United States., Vasta JD; Promega Corporation, Madison, WI, United States., Katis VL; ARUK Oxford Drug Discovery Institute, Centre for Medicines Discovery, Nuffield Department of Medicine, University of Oxford, Oxford, United Kingdom., Michaud A; Promega Corporation, Madison, WI, United States., Beck MT; Promega Corporation, Madison, WI, United States., Daglish SCD; Structural Genomics Consortium, Division of Chemical Biology and Medicinal Chemistry, Eshelman School of Pharmacy, The University of North Carolina at Chapel Hill, Chapel Hill, NC, United States., Cohen-Kedar S; Division of Gastroenterology, Rabin Medical Center, Petah-Tikva, Israel.; Felsenstein Medical Research Center, Faculty of Medical and Health Sciences, Tel-Aviv University, Tel-Aviv, Israel., Barda ES; Division of Gastroenterology, Rabin Medical Center, Petah-Tikva, Israel.; Felsenstein Medical Research Center, Faculty of Medical and Health Sciences, Tel-Aviv University, Tel-Aviv, Israel., Howell S; Structural Genomics Consortium, Division of Chemical Biology and Medicinal Chemistry, Eshelman School of Pharmacy, The University of North Carolina at Chapel Hill, Chapel Hill, NC, United States., Dotan I; Division of Gastroenterology, Rabin Medical Center, Petah-Tikva, Israel.; Felsenstein Medical Research Center, Faculty of Medical and Health Sciences, Tel-Aviv University, Tel-Aviv, Israel., Robers MB; Promega Corporation, Madison, WI, United States., Axtman AD; Structural Genomics Consortium, Division of Chemical Biology and Medicinal Chemistry, Eshelman School of Pharmacy, The University of North Carolina at Chapel Hill, Chapel Hill, NC, United States., Bashore FM; Structural Genomics Consortium, Division of Chemical Biology and Medicinal Chemistry, Eshelman School of Pharmacy, The University of North Carolina at Chapel Hill, Chapel Hill, NC, United States.
Source: Frontiers in chemical biology [Front Chem Biol] 2024; Vol. 3. Date of Electronic Publication: 2024 Jul 28.
Publication Type: Journal Article
Journal Info: Publisher: Frontiers Media S.A Country of Publication: Switzerland NLM ID: 9918716583206676 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2813-530X (Electronic) Linking ISSN: 2813530X NLM ISO Abbreviation: Front Chem Biol Subsets: PubMed not MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:2813-530X
DOI:10.3389/fchbi.2024.1447622