Structure-based design of potent pyrazolo[1,5-a]pyrimidine CDK4/6 inhibitors: biological evaluation and computational validation.

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Title: Structure-based design of potent pyrazolo[1,5-a]pyrimidine CDK4/6 inhibitors: biological evaluation and computational validation.
Authors: Binjubair FA; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University P.O. Box 2457 Riyadh 11451 Saudi Arabia., Elkotamy MS; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Alsalam University Kafr Alzayat 31611, Algharbia Egypt mahmoudelkotami@gmail.com., Mattar AA; Pharmaceutical Chemistry Department, Faculty of Pharmacy, El Saleheya El Gadida University Egypt., Almutairy BK; Department of Pharmaceutics, College of Pharmacy, Prince Sattam Bin Abdulaziz University Al-Kharj Saudi Arabia., Al-Rashood ST; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University P.O. Box 2457 Riyadh 11451 Saudi Arabia., Eldesouki MM; Scientific Research and Innovation Support Unit, Faculty of Pharmacy, Kafrelsheikh University Kafrelsheikh 33516 Egypt., Bouajila J; Laboratoire de Génie Chimique, Université de Toulouse, Toulouse INP, CNRS, LGC Toulouse France., Abdel-Aziz HA; Applied Organic Chemistry Department, National Research Centre Dokki Cairo 12622 Egypt., Fakhry MM; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Egyptian Russian University Badr City Cairo 11829 Egypt mariam-medhat@eru.edu.eg.
Source: RSC medicinal chemistry [RSC Med Chem] 2026 Apr 20. Date of Electronic Publication: 2026 Apr 20.
Publication Type: Journal Article
Journal Info: Publisher: Royal Society of Chemistry Country of Publication: England NLM ID: 101759460 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2632-8682 (Electronic) Linking ISSN: 26328682 NLM ISO Abbreviation: RSC Med Chem
Database: MEDLINE Ultimate
Description
ISSN:2632-8682
DOI:10.1039/d5md01147g