Efficacy, Structure-Activity Relationship, and Mode of Action Studies of a New Generation of Acridine/Acridone-Based Antimalarials.

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Title: Efficacy, Structure-Activity Relationship, and Mode of Action Studies of a New Generation of Acridine/Acridone-Based Antimalarials.
Authors: Maluf SEC; São Carlos Institute of Physics, University of São Paulo, São Carlos 13563-120, Brazil., Mendes GR; São Carlos Institute of Physics, University of São Paulo, São Carlos 13563-120, Brazil., Moura IMR; São Carlos Institute of Physics, University of São Paulo, São Carlos 13563-120, Brazil., de Souza GE; São Carlos Institute of Physics, University of São Paulo, São Carlos 13563-120, Brazil., Valdes TA; São Carlos Institute of Physics, University of São Paulo, São Carlos 13563-120, Brazil., Bonatto V; São Carlos Institute of Physics, University of São Paulo, São Carlos 13563-120, Brazil., Oliveira GS; São Carlos Institute of Physics, University of São Paulo, São Carlos 13563-120, Brazil., Aguiar ACC; Department of Microbiology, Immunology and Parasitology, Federal University of São Paulo, São Paulo, CEP 04023-062, Brazil., Gazarini ML; Department of Biosciences, Federal University of São Paulo, Santos 11015-020, Brazil., Puhl AC; Collaborations Pharmaceuticals, Inc., 840 Main Campus Drive, Lab 3510, Raleigh, North Carolina 27606, United States., Monakhova N; Research Center of Biotechnology RAS, 33-2 Leninsky prospect, Moscow 119071, Russia., Lepioshkin A; Research Center of Biotechnology RAS, 33-2 Leninsky prospect, Moscow 119071, Russia., Makarov V; Research Center of Biotechnology RAS, 33-2 Leninsky prospect, Moscow 119071, Russia., Lane TR; Collaborations Pharmaceuticals, Inc., 840 Main Campus Drive, Lab 3510, Raleigh, North Carolina 27606, United States., Raman R; Collaborations Pharmaceuticals, Inc., 840 Main Campus Drive, Lab 3510, Raleigh, North Carolina 27606, United States., Campolina GAS; Department of Microbiology, Immunology and Parasitology, Federal University of São Paulo, São Paulo, CEP 04023-062, Brazil., Barbosa CS; Department of Microbiology, Immunology and Parasitology, Federal University of São Paulo, São Paulo, CEP 04023-062, Brazil., Ferreira ADS; Oswaldo Cruz Foundation, Leishmaniasis and Malaria Bioassay Platform, Porto Velho 76812-245, Brazil., Teles CBG; Oswaldo Cruz Foundation, Leishmaniasis and Malaria Bioassay Platform, Porto Velho 76812-245, Brazil., Pereira DB; Research Center in Tropical Medicine of Rondônia, Porto Velho 76812-329, Brazil., Barros RRM; Department of Microbiology, Immunology and Parasitology, Federal University of São Paulo, São Paulo, CEP 04023-062, Brazil., Benavente ED; Laboratory of Experimental Cardiology, University Medical Center Utrecht, Utrecht University, Utrecht, CS 3584, The Netherlands., Ekins S; Collaborations Pharmaceuticals, Inc., 840 Main Campus Drive, Lab 3510, Raleigh, North Carolina 27606, United States., Guido RVC; São Carlos Institute of Physics, University of São Paulo, São Carlos 13563-120, Brazil.
Source: ACS infectious diseases [ACS Infect Dis] 2026 Jun 12; Vol. 12 (6), pp. 1866-1883. Date of Electronic Publication: 2026 May 25.
Publication Type: Journal Article
Journal Info: Publisher: ACS Publications Country of Publication: United States NLM ID: 101654580 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2373-8227 (Electronic) Linking ISSN: 23738227 NLM ISO Abbreviation: ACS Infect Dis Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:2373-8227
DOI:10.1021/acsinfecdis.5c00682