Nonclinical Characterization of ACP-204, a Novel Selective 5-HT2A Receptor Inverse Agonist.
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| Title: | Nonclinical Characterization of ACP-204, a Novel Selective 5-HT2A Receptor Inverse Agonist. |
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| Authors: | Burstein ES; Acadia Pharmaceuticals Inc, San Diego, California. Electronic address: eburstein@acadia-pharm.com., Olsson R; Chemical Biology and Therapeutics, Department of Experimental Medical Science, Lund University, Lund, Sweden., Skold N; RG Discovery, Lund, Sweden., Jansen KE; RG Discovery, Lund, Sweden., Azar M; Behavioral Pharma, La Jolla, California., Sandiego C; Perceptive Discovery, New Haven, Connecticut., Ridler K; Perceptive Discovery, London, United Kingdom., Rabiner EA; Perceptive Discovery, London, United Kingdom., Rhodes G; GRhodes Pharma Consulting, Los Altos, California., Dey PM; Acadia Pharmaceuticals Inc, Princeton, New Jersey., Pathak S; Acadia Pharmaceuticals Inc, Princeton, New Jersey. |
| Source: | The Journal of pharmacology and experimental therapeutics [J Pharmacol Exp Ther] 2026 Jun; Vol. 393 (6), pp. 104932. Date of Electronic Publication: 2026 May 05. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: American Society for Pharmacology and Experimental Therapeutics Country of Publication: Netherlands NLM ID: 0376362 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1521-0103 (Electronic) Linking ISSN: 00223565 NLM ISO Abbreviation: J Pharmacol Exp Ther Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 42208178 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Nonclinical Characterization of ACP-204, a Novel Selective 5-HT2A Receptor Inverse Agonist. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Burstein+ES%22">Burstein ES</searchLink>; Acadia Pharmaceuticals Inc, San Diego, California. Electronic address: eburstein@acadia-pharm.com.<br /><searchLink fieldCode="AU" term="%22Olsson+R%22">Olsson R</searchLink>; Chemical Biology and Therapeutics, Department of Experimental Medical Science, Lund University, Lund, Sweden.<br /><searchLink fieldCode="AU" term="%22Skold+N%22">Skold N</searchLink>; RG Discovery, Lund, Sweden.<br /><searchLink fieldCode="AU" term="%22Jansen+KE%22">Jansen KE</searchLink>; RG Discovery, Lund, Sweden.<br /><searchLink fieldCode="AU" term="%22Azar+M%22">Azar M</searchLink>; Behavioral Pharma, La Jolla, California.<br /><searchLink fieldCode="AU" term="%22Sandiego+C%22">Sandiego C</searchLink>; Perceptive Discovery, New Haven, Connecticut.<br /><searchLink fieldCode="AU" term="%22Ridler+K%22">Ridler K</searchLink>; Perceptive Discovery, London, United Kingdom.<br /><searchLink fieldCode="AU" term="%22Rabiner+EA%22">Rabiner EA</searchLink>; Perceptive Discovery, London, United Kingdom.<br /><searchLink fieldCode="AU" term="%22Rhodes+G%22">Rhodes G</searchLink>; GRhodes Pharma Consulting, Los Altos, California.<br /><searchLink fieldCode="AU" term="%22Dey+PM%22">Dey PM</searchLink>; Acadia Pharmaceuticals Inc, Princeton, New Jersey.<br /><searchLink fieldCode="AU" term="%22Pathak+S%22">Pathak S</searchLink>; Acadia Pharmaceuticals Inc, Princeton, New Jersey. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%220376362%22">The Journal of pharmacology and experimental therapeutics</searchLink> [J Pharmacol Exp Ther] 2026 Jun; Vol. 393 (6), pp. 104932. <i>Date of Electronic Publication: </i>2026 May 05. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22American+Society+for+Pharmacology+and+Experimental+Therapeutics%22">American Society for Pharmacology and Experimental Therapeutics </searchLink><i>Country of Publication: </i>Netherlands <i>NLM ID: </i>0376362 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1521-0103 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2200223565%22">00223565 </searchLink><i>NLM ISO Abbreviation: </i>J Pharmacol Exp Ther <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=42208178 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1016/j.jpet.2026.104932 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 104932 Titles: – TitleFull: Nonclinical Characterization of ACP-204, a Novel Selective 5-HT2A Receptor Inverse Agonist. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Burstein ES – PersonEntity: Name: NameFull: Olsson R – PersonEntity: Name: NameFull: Skold N – PersonEntity: Name: NameFull: Jansen KE – PersonEntity: Name: NameFull: Azar M – PersonEntity: Name: NameFull: Sandiego C – PersonEntity: Name: NameFull: Ridler K – PersonEntity: Name: NameFull: Rabiner EA – PersonEntity: Name: NameFull: Rhodes G – PersonEntity: Name: NameFull: Dey PM – PersonEntity: Name: NameFull: Pathak S IsPartOfRelationships: – BibEntity: Dates: – D: 01 M: 06 Text: 2026 Jun Type: published Y: 2026 Identifiers: – Type: issn-electronic Value: 1521-0103 Numbering: – Type: volume Value: 393 – Type: issue Value: 6 Titles: – TitleFull: The Journal of pharmacology and experimental therapeutics Type: main |
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