Nonclinical Characterization of ACP-204, a Novel Selective 5-HT2A Receptor Inverse Agonist.

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Title: Nonclinical Characterization of ACP-204, a Novel Selective 5-HT2A Receptor Inverse Agonist.
Authors: Burstein ES; Acadia Pharmaceuticals Inc, San Diego, California. Electronic address: eburstein@acadia-pharm.com., Olsson R; Chemical Biology and Therapeutics, Department of Experimental Medical Science, Lund University, Lund, Sweden., Skold N; RG Discovery, Lund, Sweden., Jansen KE; RG Discovery, Lund, Sweden., Azar M; Behavioral Pharma, La Jolla, California., Sandiego C; Perceptive Discovery, New Haven, Connecticut., Ridler K; Perceptive Discovery, London, United Kingdom., Rabiner EA; Perceptive Discovery, London, United Kingdom., Rhodes G; GRhodes Pharma Consulting, Los Altos, California., Dey PM; Acadia Pharmaceuticals Inc, Princeton, New Jersey., Pathak S; Acadia Pharmaceuticals Inc, Princeton, New Jersey.
Source: The Journal of pharmacology and experimental therapeutics [J Pharmacol Exp Ther] 2026 Jun; Vol. 393 (6), pp. 104932. Date of Electronic Publication: 2026 May 05.
Publication Type: Journal Article
Journal Info: Publisher: American Society for Pharmacology and Experimental Therapeutics Country of Publication: Netherlands NLM ID: 0376362 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1521-0103 (Electronic) Linking ISSN: 00223565 NLM ISO Abbreviation: J Pharmacol Exp Ther Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: Nonclinical Characterization of ACP-204, a Novel Selective 5-HT2A Receptor Inverse Agonist.
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  Data: <searchLink fieldCode="AU" term="%22Burstein+ES%22">Burstein ES</searchLink>; Acadia Pharmaceuticals Inc, San Diego, California. Electronic address: eburstein@acadia-pharm.com.<br /><searchLink fieldCode="AU" term="%22Olsson+R%22">Olsson R</searchLink>; Chemical Biology and Therapeutics, Department of Experimental Medical Science, Lund University, Lund, Sweden.<br /><searchLink fieldCode="AU" term="%22Skold+N%22">Skold N</searchLink>; RG Discovery, Lund, Sweden.<br /><searchLink fieldCode="AU" term="%22Jansen+KE%22">Jansen KE</searchLink>; RG Discovery, Lund, Sweden.<br /><searchLink fieldCode="AU" term="%22Azar+M%22">Azar M</searchLink>; Behavioral Pharma, La Jolla, California.<br /><searchLink fieldCode="AU" term="%22Sandiego+C%22">Sandiego C</searchLink>; Perceptive Discovery, New Haven, Connecticut.<br /><searchLink fieldCode="AU" term="%22Ridler+K%22">Ridler K</searchLink>; Perceptive Discovery, London, United Kingdom.<br /><searchLink fieldCode="AU" term="%22Rabiner+EA%22">Rabiner EA</searchLink>; Perceptive Discovery, London, United Kingdom.<br /><searchLink fieldCode="AU" term="%22Rhodes+G%22">Rhodes G</searchLink>; GRhodes Pharma Consulting, Los Altos, California.<br /><searchLink fieldCode="AU" term="%22Dey+PM%22">Dey PM</searchLink>; Acadia Pharmaceuticals Inc, Princeton, New Jersey.<br /><searchLink fieldCode="AU" term="%22Pathak+S%22">Pathak S</searchLink>; Acadia Pharmaceuticals Inc, Princeton, New Jersey.
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  Data: <searchLink fieldCode="JN" term="%220376362%22">The Journal of pharmacology and experimental therapeutics</searchLink> [J Pharmacol Exp Ther] 2026 Jun; Vol. 393 (6), pp. 104932. <i>Date of Electronic Publication: </i>2026 May 05.
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              Text: 2026 Jun
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