Thermodynamic profiling and fragment screening of GPCRs using grating-coupled interferometry.

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Title: Thermodynamic profiling and fragment screening of GPCRs using grating-coupled interferometry.
Authors: Churchill-Angus A; Evotec (UK) Ltd, Dorothy Crowfoot Hodgkin Campus, 95 Park Drive, Milton Park Abingdon, OX14 4RY, United Kingdom., Crespillo-Torreno S; Evotec (UK) Ltd, Dorothy Crowfoot Hodgkin Campus, 95 Park Drive, Milton Park Abingdon, OX14 4RY, United Kingdom., Griss Pascualli E; Evotec (UK) Ltd, Dorothy Crowfoot Hodgkin Campus, 95 Park Drive, Milton Park Abingdon, OX14 4RY, United Kingdom., Bertinelli M; Evotec (UK) Ltd, Dorothy Crowfoot Hodgkin Campus, 95 Park Drive, Milton Park Abingdon, OX14 4RY, United Kingdom., Grou C; Evotec (UK) Ltd, Dorothy Crowfoot Hodgkin Campus, 95 Park Drive, Milton Park Abingdon, OX14 4RY, United Kingdom., Errey JC; Evotec (UK) Ltd, Dorothy Crowfoot Hodgkin Campus, 95 Park Drive, Milton Park Abingdon, OX14 4RY, United Kingdom., Fiez-Vandal C; Evotec (UK) Ltd, Dorothy Crowfoot Hodgkin Campus, 95 Park Drive, Milton Park Abingdon, OX14 4RY, United Kingdom., Fabini E; Evotec (UK) Ltd, Dorothy Crowfoot Hodgkin Campus, 95 Park Drive, Milton Park Abingdon, OX14 4RY, United Kingdom. Electronic address: edoardo.fabini@evotec.com.
Source: SLAS discovery : advancing life sciences R & D [SLAS Discov] 2026 Sep; Vol. 42, pp. 100314. Date of Electronic Publication: 2026 Jun 04.
Publication Type: Journal Article
Journal Info: Publisher: SAGE Publications Country of Publication: United States NLM ID: 101697563 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2472-5560 (Electronic) Linking ISSN: 24725552 NLM ISO Abbreviation: SLAS Discov Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:2472-5560
DOI:10.1016/j.slasd.2026.100314