Development of a Highly Effective Bifunctional Ligand 2E-C-NETA for Targeted Lu-177 Therapy: Synthesis, Radiolabeling, In Vitro Stability, and In Vivo Biodistribution.

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Title: Development of a Highly Effective Bifunctional Ligand 2E-C-NETA for Targeted Lu-177 Therapy: Synthesis, Radiolabeling, In Vitro Stability, and In Vivo Biodistribution.
Authors: Chen Y; Department of Chemistry, Illinois Institute of Technology, Chicago, Illinois, USA., Lee Y; Department of Chemistry, Illinois Institute of Technology, Chicago, Illinois, USA., Kang CS; Department of Chemistry, Illinois Institute of Technology, Chicago, Illinois, USA., Ren S; Department of Chemistry, Illinois Institute of Technology, Chicago, Illinois, USA., Chen Y; Department of Chemistry, Illinois Institute of Technology, Chicago, Illinois, USA., Wang H; Department of Chemistry, Illinois Institute of Technology, Chicago, Illinois, USA., Bandara N; Department of Radiation Oncology, Washington University, Saint Louis, Missouri, USA., Rogers BE; Department of Radiation Oncology, Washington University, Saint Louis, Missouri, USA., Chong HS; Department of Chemistry, Illinois Institute of Technology, Chicago, Illinois, USA.
Source: ChemMedChem [ChemMedChem] 2026 Jun 15; Vol. 21 (11), pp. e70325.
Publication Type: Journal Article
Journal Info: Publisher: Wiley-VCH Country of Publication: Germany NLM ID: 101259013 Publication Model: Print Cited Medium: Internet ISSN: 1860-7187 (Electronic) Linking ISSN: 18607179 NLM ISO Abbreviation: ChemMedChem Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1860-7187
DOI:10.1002/cmdc.70325