Advances in selective inhibitors targeting the BD1 and BD2 domains of BET proteins.

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Title: Advances in selective inhibitors targeting the BD1 and BD2 domains of BET proteins.
Authors: Xie JY; Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing, 211198, China., Pang YW; Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing, 211198, China., Yu CL; Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing, 211198, China., Li YY; Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing, 211198, China. Electronic address: yuyanli@cpu.edu.cn., Shi L; Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing, 211198, China. Electronic address: shilei@cpu.edu.cn.
Source: European journal of medicinal chemistry [Eur J Med Chem] 2026 Jun 30; Vol. 317, pp. 119118. Date of Electronic Publication: 2026 Jun 30.
Publication Type: Journal Article; Review
Journal Info: Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1768-3254 (Electronic) Linking ISSN: 02235234 NLM ISO Abbreviation: Eur J Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
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DbLabel: MEDLINE Ultimate
An: 42391930
AccessLevel: 2
PubType: Academic Journal
PubTypeId: academicJournal
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  Data: Advances in selective inhibitors targeting the BD1 and BD2 domains of BET proteins.
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  Data: <searchLink fieldCode="AU" term="%22Xie+JY%22">Xie JY</searchLink>; Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing, 211198, China.<br /><searchLink fieldCode="AU" term="%22Pang+YW%22">Pang YW</searchLink>; Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing, 211198, China.<br /><searchLink fieldCode="AU" term="%22Yu+CL%22">Yu CL</searchLink>; Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing, 211198, China.<br /><searchLink fieldCode="AU" term="%22Li+YY%22">Li YY</searchLink>; Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing, 211198, China. Electronic address: yuyanli@cpu.edu.cn.<br /><searchLink fieldCode="AU" term="%22Shi+L%22">Shi L</searchLink>; Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing, 211198, China. Electronic address: shilei@cpu.edu.cn.
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  Data: <searchLink fieldCode="JN" term="%220420510%22">European journal of medicinal chemistry</searchLink> [Eur J Med Chem] 2026 Jun 30; Vol. 317, pp. 119118. <i>Date of Electronic Publication: </i>2026 Jun 30.
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  Data: Journal Article; Review
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Editions+Scientifiques+Elsevier%22">Editions Scientifiques Elsevier </searchLink><i>Country of Publication: </i>France <i>NLM ID: </i>0420510 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1768-3254 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2202235234%22">02235234 </searchLink><i>NLM ISO Abbreviation: </i>Eur J Med Chem <i>Subsets: </i>MEDLINE
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RecordInfo BibRecord:
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      – Type: doi
        Value: 10.1016/j.ejmech.2026.119118
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      – Code: eng
        Text: English
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        StartPage: 119118
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      – TitleFull: Advances in selective inhibitors targeting the BD1 and BD2 domains of BET proteins.
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            NameFull: Xie JY
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            NameFull: Pang YW
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            NameFull: Yu CL
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            NameFull: Li YY
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            – D: 30
              M: 06
              Text: 2026 Jun 30
              Type: published
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              Value: 317
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            – TitleFull: European journal of medicinal chemistry
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